XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD16-144 HeLa GCK
DTVTSELAAVkIVK
Lys1
3.1
10
uM
XMD16-144 HeLa IRAK4
DIkSANILLDEAFTAK
Lys2
-0.7
10
uM
XMD16-144 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
46.1
10
uM
XMD16-144 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
28.5
10
uM
XMD16-144 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
2.5
10
uM
XMD16-144 HeLa AMPKa1,AMPKa2
VAVkILNR
Lys1
90.9
10
uM
XMD16-144 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-2.0
10
uM
XMD16-144 HeLa DMPK
DIkPDNILLDR
Lys2
-6.6
10
uM
XMD16-144 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
0.2
10
uM
XMD16-144 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
96.5
10
uM
XMD16-144 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-3.2
10
uM
XMD16-144 HeLa CaMK2g
TSTQEYAAkIINTK
Lys1
39.3
10
uM
XMD16-144 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
83.8
10
uM
XMD16-144 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-1.3
10
uM
XMD16-144 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
-20.3
10
uM
XMD16-144 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
91.3
10
uM
XMD16-144 HeLa CDK2
DLkPQNLLINTEGAIK
Lys2
-11.0
10
uM
XMD16-144 HeLa ATR
FYIMMCkPK
ATP
-22.3
10
uM
XMD16-144 HeLa ACK
TVSVAVkCLKPDVLSQPEAMDDFIR
Lys1
79.4
10
uM
XMD16-144 HeLa CDK7
DLkPNNLLLDENGVLK
Lys2
45.8
10
uM
XMD16-144 HeLa BRAF
DLkSNNIFLHEDLTVK
Lys2
7.5
10
uM
XMD16-144 HeLa MK03
DLkPSNLLINTTCDLK
Lys2
-11.9
10
uM
XMD16-144 HeLa CaMK1a
LVAIkCIAK
Lys1
4.2
10
uM
XMD16-144 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
91.0
10
uM
XMD16-144 HeLa IRE1
DLkPHNILISMPNAHGK
Lys2
-23.3
10
uM
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