XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD16-144 | PC-3 | MK03 | DLkPSNLLINTTCDLK | Lys2 | 14.5 | 10 | uM |
| XMD16-144 | PC-3 | FYN,SRC,YES | QGAkFPIKWTAPEAALYGR | Activation Loop | 66.9 | 10 | uM |
| XMD16-144 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -3.6 | 10 | uM |
| XMD16-144 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 4.4 | 10 | uM |
| XMD16-144 | PC-3 | FER | TSVAVkTCKEDLPQELK | Lys1 | 51.1 | 10 | uM |
| XMD16-144 | PC-3 | AMPKa1,AMPKa2 | VAVkILNR | Lys1 | 91.3 | 10 | uM |
| XMD16-144 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 13.9 | 10 | uM |
| XMD16-144 | PC-3 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 73.5 | 10 | uM |
| XMD16-144 | PC-3 | EGFR | IPVAIkELR | Lys1 | 3.7 | 10 | uM |
| XMD16-144 | PC-3 | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 93.6 | 10 | uM |
| XMD16-144 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -17.8 | 10 | uM |
| XMD16-144 | PC-3 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIkTCK | Lys1 | 80.3 | 10 | uM |
| XMD16-144 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 47.3 | 10 | uM |
| XMD16-144 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | 26.8 | 10 | uM |
| XMD16-144 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | 49.2 | 10 | uM |
| XMD16-144 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 16.6 | 10 | uM |
| XMD16-144 | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 82.5 | 10 | uM |
| XMD16-144 | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 5.9 | 10 | uM |
| XMD16-144 | PC-3 | CDK5 | NRETHEIVALkR | Lys1 | -1.9 | 10 | uM |
| XMD16-144 | PC-3 | ATR | FYIMMCkPK | ATP | -16.0 | 10 | uM |
| XMD16-144 | PC-3 | CDK9 | DMkAANVLITR | Lys2 | -34.5 | 10 | uM |
| XMD16-144 | PC-3 | CHK2 | VAIkIISK | Lys1 | 49.6 | 10 | uM |
| XMD16-144 | PC-3 | KC1A | DIkPDNFLMGIGR | Lys2 | -16.6 | 10 | uM |
| XMD16-144 | PC-3 | CK1d,CK1e | DVkPDNFLMGLGKK | Lys2 | -12.3 | 10 | uM |
| XMD16-144 | PC-3 | GCN2_domain2 | DLkPVNIFLDSDDHVK | Lys2 | -4.6 | 10 | uM |