Evaluation of the sensitivities of six triple-negative breast cancer (TNBC) cell lines to 23 different PI3K/AKT/mTOR inhibitors or to a MEK inhibitor (trametinib). Dataset 1 of 2: GR values. - Dataset (ID:20364)
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Cell line | Drug name | Experimental replicate | Timepoint | Drug concentration | Live cell count | Average live cell count, DMSO control | Average live cell count (time = 0) | Log10(drug concentration) | GR value | Relative cell count (treatment versus DMSO) | Cell doublings (DMSO control) | Experiment name |
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HCC70 | WYE-125132 | 2 | 72 | 1.0 | 1402.5 | 2308.5 | 722.8 | 0.0 | 0.485 | 0.608 | 1.675 | HCC70 WYE125132 0 2 72 |
HCC70 | WYE-125132 | 2 | 72 | 0.001 | 2297.5 | 2308.5 | 722.8 | -3.0 | 0.994 | 0.995 | 1.675 | HCC70 WYE125132 0 2 72 |
HCC70 | WYE-125132 | 2 | 72 | 0.32 | 1397.0 | 2308.5 | 722.8 | -0.495 | 0.482 | 0.605 | 1.675 | HCC70 WYE125132 0 2 72 |
HCC70 | WYE-125132 | 2 | 72 | 0.1 | 1462.3 | 2308.5 | 722.8 | -1.0 | 0.523 | 0.633 | 1.675 | HCC70 WYE125132 0 2 72 |
HCC70 | WYE-125132 | 2 | 72 | 3.2 | 1379.5 | 2308.5 | 722.8 | 0.505 | 0.471 | 0.598 | 1.675 | HCC70 WYE125132 0 2 72 |
HCC70 | WYE-125132 | 2 | 72 | 0.0032 | 2162.8 | 2308.5 | 722.8 | -2.49 | 0.924 | 0.937 | 1.675 | HCC70 WYE125132 0 2 72 |
HCC70 | WYE-125132 | 2 | 72 | 0.032 | 1724.8 | 2308.5 | 722.8 | -1.49 | 0.681 | 0.747 | 1.675 | HCC70 WYE125132 0 2 72 |
HCC70 | WYE-125132 | 2 | 72 | 0.01 | 2029.3 | 2308.5 | 722.8 | -2.0 | 0.852 | 0.879 | 1.675 | HCC70 WYE125132 0 2 72 |
HCC70 | GDC-0980 | 2 | 72 | 0.32 | 1350.5 | 2310.0 | 722.8 | -0.495 | 0.452 | 0.585 | 1.676 | HCC70 GDC0980 0 2 72 |
HCC70 | GDC-0980 | 2 | 72 | 0.032 | 2236.5 | 2310.0 | 722.8 | -1.49 | 0.962 | 0.968 | 1.676 | HCC70 GDC0980 0 2 72 |
HCC70 | GDC-0980 | 2 | 72 | 0.0032 | 2472.8 | 2310.0 | 722.8 | -2.49 | 1.080 | 1.070 | 1.676 | HCC70 GDC0980 0 2 72 |
HCC70 | GDC-0980 | 2 | 72 | 3.2 | 623.0 | 2310.0 | 722.8 | 0.505 | -0.085 | 0.270 | 1.676 | HCC70 GDC0980 0 2 72 |
HCC70 | GDC-0980 | 2 | 72 | 1.0 | 1043.3 | 2310.0 | 722.8 | 0.0 | 0.245 | 0.452 | 1.676 | HCC70 GDC0980 0 2 72 |
HCC70 | GDC-0980 | 2 | 72 | 0.1 | 1822.5 | 2310.0 | 722.8 | -1.0 | 0.736 | 0.789 | 1.676 | HCC70 GDC0980 0 2 72 |
HCC70 | GDC-0980 | 2 | 72 | 0.001 | 2471.0 | 2310.0 | 722.8 | -3.0 | 1.080 | 1.070 | 1.676 | HCC70 GDC0980 0 2 72 |
HCC70 | GDC-0980 | 2 | 72 | 0.01 | 2388.0 | 2310.0 | 722.8 | -2.0 | 1.040 | 1.030 | 1.676 | HCC70 GDC0980 0 2 72 |
HCC70 | Dactolisib | 2 | 72 | 1.0 | 1321.3 | 2310.8 | 722.8 | 0.0 | 0.433 | 0.572 | 1.677 | HCC70 BEZ235 0 2 72 |
HCC70 | Dactolisib | 2 | 72 | 0.032 | 1708.0 | 2310.8 | 722.8 | -1.49 | 0.670 | 0.739 | 1.677 | HCC70 BEZ235 0 2 72 |
HCC70 | Dactolisib | 2 | 72 | 0.0032 | 2137.3 | 2310.8 | 722.8 | -2.49 | 0.909 | 0.925 | 1.677 | HCC70 BEZ235 0 2 72 |
HCC70 | Dactolisib | 2 | 72 | 0.1 | 1557.0 | 2310.8 | 722.8 | -1.0 | 0.580 | 0.674 | 1.677 | HCC70 BEZ235 0 2 72 |
HCC70 | Dactolisib | 2 | 72 | 3.2 | 1033.3 | 2310.8 | 722.8 | 0.505 | 0.238 | 0.447 | 1.677 | HCC70 BEZ235 0 2 72 |
HCC70 | Dactolisib | 2 | 72 | 0.01 | 2010.0 | 2310.8 | 722.8 | -2.0 | 0.840 | 0.870 | 1.677 | HCC70 BEZ235 0 2 72 |
HCC70 | Dactolisib | 2 | 72 | 0.001 | 2350.5 | 2310.8 | 722.8 | -3.0 | 1.020 | 1.020 | 1.677 | HCC70 BEZ235 0 2 72 |
HCC70 | Dactolisib | 2 | 72 | 0.32 | 1509.8 | 2310.8 | 722.8 | -0.495 | 0.552 | 0.653 | 1.677 | HCC70 BEZ235 0 2 72 |
HCC70 | Omipalisib | 2 | 72 | 0.32 | 281.3 | 2319.3 | 722.8 | -0.495 | -0.429 | 0.121 | 1.682 | HCC70 GSK458 0 2 72 |