Breast Cancer Deubiquitinating Enzyme (DUB) Inhibitor Profiling: Fixed-cell GR measures of 21 breast cell lines to 32 small molecule perturbagens. Dataset 1 of 2: Normalized growth rate inhibition values. - Dataset (ID:20350)

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Cell Small Molecule Small Mol Concentration (uM) Mean Normalized Growth Rate Inhibition (GR) Value Increased Fraction Dead
HCC1500 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one
3.16
0.9490 -0.01482
HCC1500 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one
9.992797406
1.0427 0.01003
HCC1500 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one
31.6
1.0783 -0.01719
HCC1500 5-(4-fluorophenyl)-3-hydroxy-4-(5-methyl-2-furoyl)-1-(3-pyridinylmethyl)-1,5-dihydro-2H-pyrrol-2-one
50.0
1.1258 0.00322
HCC1500 SB1-F-21
0.009992797
1.1254 -0.02192
HCC1500 SB1-F-21
0.0316
1.0976 0.03144
HCC1500 SB1-F-21
0.099927974
0.8251 0.06376
HCC1500 SB1-F-21
0.316
0.5060 0.21325
HCC1500 SB1-F-21
0.999279741
-0.2777 0.53698
HCC1500 SB1-F-21
3.16
-0.4645 0.58223
HCC1500 SB1-F-21
9.992797406
-0.3661 0.55388
HCC1500 SB1-F-21
31.6
-0.4475 0.54989
HCC1500 SB1-F-21
50.0
-0.4684 0.32988
HCC1500 SB1-F-22
0.009992797
1.0837 0.00619
HCC1500 SB1-F-22
0.0316
1.0584 0.02251
HCC1500 SB1-F-22
0.099927974
1.1421 0.02415
HCC1500 SB1-F-22
0.316
0.9485 0.04596
HCC1500 SB1-F-22
0.999279741
0.7937 0.03090
HCC1500 SB1-F-22
3.16
0.7744 0.06866
HCC1500 SB1-F-22
9.992797406
0.5383 0.18864
HCC1500 SB1-F-22
31.6
0.0425 0.35773
HCC1500 SB1-F-22
50.0
0.2075 0.09658
HCC1500 SJB2-043
0.00316
0.9407 -0.00346
HCC1500 SJB2-043
0.009992797
0.9523 0.00765
HCC1500 SJB2-043
0.0316
1.0268 0.03184