Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 2 of 2: Calculated dose response metrics - Dataset (ID:20344)
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Cell | Small Molecule | Primary Target | Pathway | GR50 | GRmax | GR_AOC | Death_AUC | GR Hill Coefficient | GEC50 | GR r2 |
---|---|---|---|---|---|---|---|---|---|---|
MDA-MB-468 | Volasertib | PLK | Cell cycle | 0.002104 | -0.4485 | 0.9279 | 0.3934 | 2.9173 | 0.0026072 | 0.99938 |
PDX1258 | Taxol | Chemo | Chemotherapy | 0.0021522 | -0.0818 | 0.6797 | 0.2357 | 1.2501 | 0.0022935 | 0.98829 |
CAMA-1 | Taxol | Chemo | Chemotherapy | 0.0022699 | -0.4944 | 0.9525 | 0.3547 | 2.4920 | 0.0029769 | 0.99478 |
SK-BR-3 | Luminespib | HSP90 | Misc | 0.0022783 | -0.0766 | 0.7140 | 0.1099 | 2.5203 | 0.0024311 | 0.9977 |
MDA-MB-231 | Taxol | Chemo | Chemotherapy | 0.0023185 | -0.1204 | 0.7021 | 0.2576 | 1.1720 | 0.0026636 | 0.96432 |
MDA-MB-453 | Taxol | Chemo | Chemotherapy | 0.002374 | 0.0356 | 0.6674 | 0.1683 | 1.2620 | 0.0023576 | 0.81734 |
PDX1328 | Luminespib | HSP90 | Misc | 0.0023764 | -0.4697 | 0.8697 | 0.1444 | 1.9222 | 0.0032941 | 0.9864 |
HCC1937 | Taxol | Chemo | Chemotherapy | 0.0024514 | 0.0104 | 0.6576 | 0.2104 | 2.2541 | 0.0024561 | 0.99541 |
SUM1315MO2 | Taxol | Chemo | Chemotherapy | 0.0024623 | -0.3258 | 0.7931 | 0.2940 | 2.0093 | 0.0030737 | 0.99498 |
HCC1954 | Taxol | Chemo | Chemotherapy | 0.0024667 | -0.3961 | 0.8347 | 0.4142 | 1.6514 | 0.0034177 | 0.98666 |
PDXHCI002 | Taxol | Chemo | Chemotherapy | 0.0024935 | -0.5117 | 0.9207 | 0.3881 | 2.7479 | 0.0031656 | 0.99139 |
PDX1328 | Volasertib | PLK | Cell cycle | 0.0025124 | -0.5731 | 0.9694 | 0.2182 | 2.8453 | 0.0032751 | 0.99856 |
HCC1395 | Everolimus | mTOR1 | PI3K/mTOR | 0.0025601 | 0.4042 | 0.5551 | 0.0370 | 0.4448 | 5.3346e-05 | 0.76727 |
Hs 578T | Volasertib | PLK | Cell cycle | 0.0025675 | -0.3123 | 0.8198 | 0.3337 | 3.0081 | 0.0029864 | 0.9987 |
MDA-MB-231 | Trametinib | MEK | MAPK/nRTK | 0.0026306 | -0.1785 | 0.7224 | 0.2816 | 1.1618 | 0.0033911 | 0.99829 |
SK-BR-3 | INK-128 | mTORC1/2 | PI3K/mTOR | 0.0026508 | -0.5064 | 0.9712 | 0.2693 | 1.0983 | 0.0044617 | 0.98817 |
MCF 10A | Taxol | Chemo | Chemotherapy | 0.0026843 | -0.1256 | 0.7023 | 0.2576 | 1.8234 | 0.003018 | 0.9967 |
MCF7 | Everolimus | mTOR1 | PI3K/mTOR | 0.0026919 | 0.3865 | 0.5643 | 0.0341 | 0.2603 | 1.8439e-05 | 0.90097 |
MDA-MB-134-VI | Volasertib | PLK | Cell cycle | 0.0027209 | -0.6274 | 1.0260 | 0.2671 | 5.0000 | 0.0032225 | 0.99553 |
BT-549 | Taxol | Chemo | Chemotherapy | 0.0027257 | -0.2074 | 0.6989 | 0.2304 | 1.9420 | 0.0030953 | 0.98743 |
CAL-85-1 | Taxol | Chemo | Chemotherapy | 0.0027273 | -0.3464 | 0.7931 | 0.3351 | 2.0210 | 0.0033785 | 0.95638 |
HCC1395 | Topotecan | Topo I | Chemotherapy | 0.0027504 | -0.5835 | 1.0761 | 0.3115 | 0.5889 | 0.0088299 | 0.93292 |
HCC1806 | Volasertib | PLK | Cell cycle | 0.0027998 | -0.1323 | 0.7262 | 0.2950 | 5.0000 | 0.0029495 | 0.99776 |
CAL-120 | Luminespib | HSP90 | Misc | 0.0028134 | -0.1149 | 0.6933 | 0.1709 | 1.6073 | 0.0031386 | 0.99357 |
HCC1428 | Luminespib | HSP90 | Misc | 0.0028629 | -0.0043 | 0.6375 | 0.0972 | 5.0000 | 0.0028677 | 0.99886 |