Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
HCC1806 | Neratinib | 0.1 | EGFR/HER2 | RTK | 0.7682 | 0.05014 |
HCC1806 | Tivantinib | 0.1 | MET | RTK | 0.9630 | 0.00521 |
HCC1806 | Ceritinib | 1.0 | ALK | RTK | 0.8590 | 0.02331 |
HCC1806 | Neratinib | 0.031623 | EGFR/HER2 | RTK | 0.8990 | 0.02920 |
HCC1806 | Tivantinib | 0.001 | MET | RTK | 1.0293 | 0.00356 |
HCC1806 | Tivantinib | 0.031623 | MET | RTK | 1.0186 | 0.00130 |
HCC1806 | Ceritinib | 0.01 | ALK | RTK | 1.0487 | 0.00015 |
HCC1806 | Ceritinib | 0.31623 | ALK | RTK | 1.1237 | -0.00775 |
HCC1806 | Neratinib | 0.00031623 | EGFR/HER2 | RTK | 1.0684 | 0.00476 |
HCC1806 | Neratinib | 0.01 | EGFR/HER2 | RTK | 0.9959 | 0.01677 |
HCC1806 | Neratinib | 1.0 | EGFR/HER2 | RTK | 0.5513 | 0.07881 |
HCC1806 | Neratinib | 3.1623 | EGFR/HER2 | RTK | -0.0883 | 0.43583 |
HCC1806 | Tivantinib | 0.0031623 | MET | RTK | 0.9997 | 0.00401 |
HCC1806 | Tivantinib | 0.01 | MET | RTK | 1.0496 | -0.00152 |
HCC1806 | Ceritinib | 0.001 | ALK | RTK | 1.0121 | 0.00605 |
HCC1806 | Ceritinib | 0.0031623 | ALK | RTK | 1.0658 | -0.00214 |
HCC1806 | Ceritinib | 0.031623 | ALK | RTK | 1.0774 | -0.00516 |
HCC1806 | Ceritinib | 0.1 | ALK | RTK | 1.0986 | -0.00400 |
HCC1806 | Ceritinib | 3.1623 | ALK | RTK | 0.1763 | 0.12321 |
HCC1806 | Ceritinib | 10.0 | ALK | RTK | -0.4060 | 0.58043 |
HCC1806 | Neratinib | 0.001 | EGFR/HER2 | RTK | 1.0533 | -0.00088 |
HCC1806 | Neratinib | 0.0031623 | EGFR/HER2 | RTK | 1.0102 | 0.00509 |
HCC1806 | Neratinib | 0.31623 | EGFR/HER2 | RTK | 0.7026 | 0.06151 |
HCC1806 | Tivantinib | 1.0 | MET | RTK | -0.1778 | 0.49866 |
HCC1806 | Tivantinib | 0.31623 | MET | RTK | 0.3568 | 0.15622 |