Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)

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Cell Small Molecule Small Mol Concentration (uM) Primary Target Pathway Mean Normalized Growth Rate Inhibition Value Increased Fraction Dead
HCC1806 Neratinib
0.1
EGFR/HER2
RTK
0.7682 0.05014
HCC1806 Tivantinib
0.1
MET
RTK
0.9630 0.00521
HCC1806 Ceritinib
1.0
ALK
RTK
0.8590 0.02331
HCC1806 Neratinib
0.031623
EGFR/HER2
RTK
0.8990 0.02920
HCC1806 Tivantinib
0.001
MET
RTK
1.0293 0.00356
HCC1806 Tivantinib
0.031623
MET
RTK
1.0186 0.00130
HCC1806 Ceritinib
0.01
ALK
RTK
1.0487 0.00015
HCC1806 Ceritinib
0.31623
ALK
RTK
1.1237 -0.00775
HCC1806 Neratinib
0.00031623
EGFR/HER2
RTK
1.0684 0.00476
HCC1806 Neratinib
0.01
EGFR/HER2
RTK
0.9959 0.01677
HCC1806 Neratinib
1.0
EGFR/HER2
RTK
0.5513 0.07881
HCC1806 Neratinib
3.1623
EGFR/HER2
RTK
-0.0883 0.43583
HCC1806 Tivantinib
0.0031623
MET
RTK
0.9997 0.00401
HCC1806 Tivantinib
0.01
MET
RTK
1.0496 -0.00152
HCC1806 Ceritinib
0.001
ALK
RTK
1.0121 0.00605
HCC1806 Ceritinib
0.0031623
ALK
RTK
1.0658 -0.00214
HCC1806 Ceritinib
0.031623
ALK
RTK
1.0774 -0.00516
HCC1806 Ceritinib
0.1
ALK
RTK
1.0986 -0.00400
HCC1806 Ceritinib
3.1623
ALK
RTK
0.1763 0.12321
HCC1806 Ceritinib
10.0
ALK
RTK
-0.4060 0.58043
HCC1806 Neratinib
0.001
EGFR/HER2
RTK
1.0533 -0.00088
HCC1806 Neratinib
0.0031623
EGFR/HER2
RTK
1.0102 0.00509
HCC1806 Neratinib
0.31623
EGFR/HER2
RTK
0.7026 0.06151
HCC1806 Tivantinib
1.0
MET
RTK
-0.1778 0.49866
HCC1806 Tivantinib
0.31623
MET
RTK
0.3568 0.15622
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