Breast Cancer Profiling Project, Drug Sensitivity phase I: Fixed-cell GR measures of 35 breast cell lines to 34 small molecule perturbagens from library plate I. Dataset 1 of 2: Normalized growth rate inhibition values - Dataset (ID:20343)
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Cell | Small Molecule | Small Mol Concentration (uM) | Primary Target | Pathway | Mean Normalized Growth Rate Inhibition Value | Increased Fraction Dead |
---|---|---|---|---|---|---|
HME1 | Tivantinib | 0.1 | MET | RTK | 0.0360 | 0.28655 |
HME1 | Tivantinib | 0.31623 | MET | RTK | -0.1213 | 0.32977 |
HME1 | Tivantinib | 1.0 | MET | RTK | -0.1181 | 0.36459 |
HME1 | Tivantinib | 3.1623 | MET | RTK | -0.1308 | 0.42862 |
HME1 | Tivantinib | 10.0 | MET | RTK | -0.1612 | 0.44114 |
HME1 | Cediranib | 0.001 | VEGFR/cKIT | RTK | 1.0678 | 0.00264 |
HME1 | Cediranib | 0.0031623 | VEGFR/cKIT | RTK | 1.0942 | 0.00158 |
HME1 | Cediranib | 0.01 | VEGFR/cKIT | RTK | 1.0882 | 0.00363 |
HME1 | Cediranib | 0.031623 | VEGFR/cKIT | RTK | 1.1129 | -0.00121 |
HME1 | Cediranib | 0.1 | VEGFR/cKIT | RTK | 1.1080 | 0.00358 |
HME1 | Cediranib | 0.31623 | VEGFR/cKIT | RTK | 1.0962 | 0.00312 |
HME1 | Cediranib | 1.0 | VEGFR/cKIT | RTK | 1.1291 | 0.00336 |
HME1 | Cediranib | 3.1623 | VEGFR/cKIT | RTK | 0.9898 | 0.00021 |
HME1 | Cediranib | 10.0 | VEGFR/cKIT | RTK | 0.0275 | 0.20231 |
HME1 | Cabozantinib | 0.001 | VEGFR2/MET | RTK | 1.0351 | 0.00073 |
HME1 | Cabozantinib | 0.0031623 | VEGFR2/MET | RTK | 1.0834 | 0.00218 |
HME1 | Cabozantinib | 0.01 | VEGFR2/MET | RTK | 1.0751 | 0.00001 |
HME1 | Cabozantinib | 0.031623 | VEGFR2/MET | RTK | 1.0964 | 0.00018 |
HME1 | Cabozantinib | 0.1 | VEGFR2/MET | RTK | 1.0687 | 0.00256 |
HME1 | Cabozantinib | 0.31623 | VEGFR2/MET | RTK | 1.0399 | 0.01058 |
HME1 | Cabozantinib | 1.0 | VEGFR2/MET | RTK | 0.9599 | 0.00869 |
HME1 | Cabozantinib | 3.1623 | VEGFR2/MET | RTK | 0.5190 | 0.02233 |
HME1 | Cabozantinib | 10.0 | VEGFR2/MET | RTK | -0.1052 | 0.18653 |
SUM1315MO2 | Abemaciclib | 0.001 | CDK4/6 | Cell cycle | 1.0408 | 0.00466 |
SUM1315MO2 | Abemaciclib | 0.0031623 | CDK4/6 | Cell cycle | 0.7932 | 0.00034 |