Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib INSR 85.0 100
nM
Taselisib INSR 100.0 1000
nM
Taselisib INSRR 100.0 100
nM
Taselisib INSRR 100.0 1000
nM
Taselisib IRAK1 87.0 100
nM
Taselisib IRAK1 100.0 1000
nM
Taselisib IRAK3 93.0 100
nM
Taselisib IRAK3 99.0 1000
nM
Taselisib IRAK4 100.0 100
nM
Taselisib IRAK4 100.0 1000
nM
Taselisib ITK 98.0 100
nM
Taselisib ITK 100.0 1000
nM
Taselisib JAK1(JH1domain-catalytic) 90.0 100
nM
Taselisib JAK1(JH1domain-catalytic) 94.0 1000
nM
Taselisib JAK1(JH2domain-pseudokinase) 95.0 100
nM
Taselisib JAK1(JH2domain-pseudokinase) 94.0 1000
nM
Taselisib JAK2(JH1domain-catalytic) 75.0 100
nM
Taselisib JAK2(JH1domain-catalytic) 89.0 1000
nM
Taselisib JAK3(JH1domain-catalytic) 90.0 100
nM
Taselisib JAK3(JH1domain-catalytic) 100.0 1000
nM
Taselisib JNK1 100.0 100
nM
Taselisib JNK1 88.0 1000
nM
Taselisib MK09 97.0 100
nM
Taselisib MK09 97.0 1000
nM
Taselisib JNK3 100.0 100
nM