Taselisib KINOMEscan - Dataset (ID:20264)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Taselisib | INSR | 85.0 | 100 | nM |
Taselisib | INSR | 100.0 | 1000 | nM |
Taselisib | INSRR | 100.0 | 100 | nM |
Taselisib | INSRR | 100.0 | 1000 | nM |
Taselisib | IRAK1 | 87.0 | 100 | nM |
Taselisib | IRAK1 | 100.0 | 1000 | nM |
Taselisib | IRAK3 | 93.0 | 100 | nM |
Taselisib | IRAK3 | 99.0 | 1000 | nM |
Taselisib | IRAK4 | 100.0 | 100 | nM |
Taselisib | IRAK4 | 100.0 | 1000 | nM |
Taselisib | ITK | 98.0 | 100 | nM |
Taselisib | ITK | 100.0 | 1000 | nM |
Taselisib | JAK1(JH1domain-catalytic) | 90.0 | 100 | nM |
Taselisib | JAK1(JH1domain-catalytic) | 94.0 | 1000 | nM |
Taselisib | JAK1(JH2domain-pseudokinase) | 95.0 | 100 | nM |
Taselisib | JAK1(JH2domain-pseudokinase) | 94.0 | 1000 | nM |
Taselisib | JAK2(JH1domain-catalytic) | 75.0 | 100 | nM |
Taselisib | JAK2(JH1domain-catalytic) | 89.0 | 1000 | nM |
Taselisib | JAK3(JH1domain-catalytic) | 90.0 | 100 | nM |
Taselisib | JAK3(JH1domain-catalytic) | 100.0 | 1000 | nM |
Taselisib | JNK1 | 100.0 | 100 | nM |
Taselisib | JNK1 | 88.0 | 1000 | nM |
Taselisib | MK09 | 97.0 | 100 | nM |
Taselisib | MK09 | 97.0 | 1000 | nM |
Taselisib | JNK3 | 100.0 | 100 | nM |