Taselisib KINOMEscan - Dataset (ID:20264)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Taselisib | CDK7 | 92.0 | 100 | nM |
Taselisib | CDK7 | 96.0 | 1000 | nM |
Taselisib | CDK8 | 97.0 | 100 | nM |
Taselisib | CDK8 | 89.0 | 1000 | nM |
Taselisib | CDK9 | 100.0 | 100 | nM |
Taselisib | CDK9 | 100.0 | 1000 | nM |
Taselisib | CDKL1 | 71.0 | 100 | nM |
Taselisib | CDKL1 | 87.0 | 1000 | nM |
Taselisib | CDKL2 | 93.0 | 100 | nM |
Taselisib | CDKL2 | 85.0 | 1000 | nM |
Taselisib | CDKL3 | 88.0 | 100 | nM |
Taselisib | CDKL3 | 93.0 | 1000 | nM |
Taselisib | CDKL5 | 99.0 | 100 | nM |
Taselisib | CDKL5 | 95.0 | 1000 | nM |
Taselisib | CHEK1 | 99.0 | 100 | nM |
Taselisib | CHEK1 | 100.0 | 1000 | nM |
Taselisib | CHK2 | 100.0 | 100 | nM |
Taselisib | CHK2 | 100.0 | 1000 | nM |
Taselisib | CIT | 88.0 | 100 | nM |
Taselisib | CIT | 97.0 | 1000 | nM |
Taselisib | CLK1 | 92.0 | 100 | nM |
Taselisib | CLK1 | 94.0 | 1000 | nM |
Taselisib | CLK2 | 88.0 | 100 | nM |
Taselisib | CLK2 | 100.0 | 1000 | nM |
Taselisib | CLK3 | 91.0 | 100 | nM |