Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib CDK7 92.0 100
nM
Taselisib CDK7 96.0 1000
nM
Taselisib CDK8 97.0 100
nM
Taselisib CDK8 89.0 1000
nM
Taselisib CDK9 100.0 100
nM
Taselisib CDK9 100.0 1000
nM
Taselisib CDKL1 71.0 100
nM
Taselisib CDKL1 87.0 1000
nM
Taselisib CDKL2 93.0 100
nM
Taselisib CDKL2 85.0 1000
nM
Taselisib CDKL3 88.0 100
nM
Taselisib CDKL3 93.0 1000
nM
Taselisib CDKL5 99.0 100
nM
Taselisib CDKL5 95.0 1000
nM
Taselisib CHEK1 99.0 100
nM
Taselisib CHEK1 100.0 1000
nM
Taselisib CHK2 100.0 100
nM
Taselisib CHK2 100.0 1000
nM
Taselisib CIT 88.0 100
nM
Taselisib CIT 97.0 1000
nM
Taselisib CLK1 92.0 100
nM
Taselisib CLK1 94.0 1000
nM
Taselisib CLK2 88.0 100
nM
Taselisib CLK2 100.0 1000
nM
Taselisib CLK3 91.0 100
nM