Taselisib KINOMEscan - Dataset (ID:20264)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Taselisib | JNK3 | 97.0 | 1000 | nM |
Taselisib | KIT | 100.0 | 100 | nM |
Taselisib | KIT | 100.0 | 1000 | nM |
Taselisib | KIT(A829P) | 100.0 | 100 | nM |
Taselisib | KIT(A829P) | 100.0 | 1000 | nM |
Taselisib | KIT(D816H) | 100.0 | 100 | nM |
Taselisib | KIT(D816H) | 95.0 | 1000 | nM |
Taselisib | KIT(D816V) | 97.0 | 100 | nM |
Taselisib | KIT(D816V) | 100.0 | 1000 | nM |
Taselisib | KIT(L576P) | 100.0 | 100 | nM |
Taselisib | KIT(L576P) | 88.0 | 1000 | nM |
Taselisib | KIT(V559D) | 100.0 | 100 | nM |
Taselisib | KIT(V559D) | 97.0 | 1000 | nM |
Taselisib | KIT(V559D,T670I) | 100.0 | 100 | nM |
Taselisib | KIT(V559D,T670I) | 100.0 | 1000 | nM |
Taselisib | KIT(V559D,V654A) | 100.0 | 100 | nM |
Taselisib | KIT(V559D,V654A) | 100.0 | 1000 | nM |
Taselisib | KIT-autoinhibited | 84.0 | 100 | nM |
Taselisib | KIT-autoinhibited | 98.0 | 1000 | nM |
Taselisib | LATS1 | 100.0 | 100 | nM |
Taselisib | LATS1 | 66.0 | 1000 | nM |
Taselisib | LATS2 | 84.0 | 100 | nM |
Taselisib | LATS2 | 100.0 | 1000 | nM |
Taselisib | LCK | 94.0 | 100 | nM |
Taselisib | LCK | 90.0 | 1000 | nM |