Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib JNK3 97.0 1000
nM
Taselisib KIT 100.0 100
nM
Taselisib KIT 100.0 1000
nM
Taselisib KIT(A829P) 100.0 100
nM
Taselisib KIT(A829P) 100.0 1000
nM
Taselisib KIT(D816H) 100.0 100
nM
Taselisib KIT(D816H) 95.0 1000
nM
Taselisib KIT(D816V) 97.0 100
nM
Taselisib KIT(D816V) 100.0 1000
nM
Taselisib KIT(L576P) 100.0 100
nM
Taselisib KIT(L576P) 88.0 1000
nM
Taselisib KIT(V559D) 100.0 100
nM
Taselisib KIT(V559D) 97.0 1000
nM
Taselisib KIT(V559D,T670I) 100.0 100
nM
Taselisib KIT(V559D,T670I) 100.0 1000
nM
Taselisib KIT(V559D,V654A) 100.0 100
nM
Taselisib KIT(V559D,V654A) 100.0 1000
nM
Taselisib KIT-autoinhibited 84.0 100
nM
Taselisib KIT-autoinhibited 98.0 1000
nM
Taselisib LATS1 100.0 100
nM
Taselisib LATS1 66.0 1000
nM
Taselisib LATS2 84.0 100
nM
Taselisib LATS2 100.0 1000
nM
Taselisib LCK 94.0 100
nM
Taselisib LCK 90.0 1000
nM