Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib MAST1 67.0 100
nM
Taselisib MAST1 69.0 1000
nM
Taselisib MP2K1 81.0 100
nM
Taselisib MP2K1 89.0 1000
nM
Taselisib MP2K2 85.0 100
nM
Taselisib MP2K2 92.0 1000
nM
Taselisib MP2K3 77.0 100
nM
Taselisib MP2K3 97.0 1000
nM
Taselisib MP2K4 100.0 100
nM
Taselisib MP2K4 89.0 1000
nM
Taselisib MP2K5 100.0 100
nM
Taselisib MP2K5 95.0 1000
nM
Taselisib MP2K6 100.0 100
nM
Taselisib MP2K6 100.0 1000
nM
Taselisib MELK 91.0 100
nM
Taselisib MELK 100.0 1000
nM
Taselisib MERTK 95.0 100
nM
Taselisib MERTK 75.0 1000
nM
Taselisib MET 85.0 100
nM
Taselisib MET 100.0 1000
nM
Taselisib MET(M1250T) 92.0 100
nM
Taselisib MET(M1250T) 93.0 1000
nM
Taselisib MET(Y1235D) 89.0 100
nM
Taselisib MET(Y1235D) 79.0 1000
nM
Taselisib MINK 88.0 100
nM