Taselisib KINOMEscan - Dataset (ID:20264)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Taselisib | MAST1 | 67.0 | 100 | nM |
Taselisib | MAST1 | 69.0 | 1000 | nM |
Taselisib | MP2K1 | 81.0 | 100 | nM |
Taselisib | MP2K1 | 89.0 | 1000 | nM |
Taselisib | MP2K2 | 85.0 | 100 | nM |
Taselisib | MP2K2 | 92.0 | 1000 | nM |
Taselisib | MP2K3 | 77.0 | 100 | nM |
Taselisib | MP2K3 | 97.0 | 1000 | nM |
Taselisib | MP2K4 | 100.0 | 100 | nM |
Taselisib | MP2K4 | 89.0 | 1000 | nM |
Taselisib | MP2K5 | 100.0 | 100 | nM |
Taselisib | MP2K5 | 95.0 | 1000 | nM |
Taselisib | MP2K6 | 100.0 | 100 | nM |
Taselisib | MP2K6 | 100.0 | 1000 | nM |
Taselisib | MELK | 91.0 | 100 | nM |
Taselisib | MELK | 100.0 | 1000 | nM |
Taselisib | MERTK | 95.0 | 100 | nM |
Taselisib | MERTK | 75.0 | 1000 | nM |
Taselisib | MET | 85.0 | 100 | nM |
Taselisib | MET | 100.0 | 1000 | nM |
Taselisib | MET(M1250T) | 92.0 | 100 | nM |
Taselisib | MET(M1250T) | 93.0 | 1000 | nM |
Taselisib | MET(Y1235D) | 89.0 | 100 | nM |
Taselisib | MET(Y1235D) | 79.0 | 1000 | nM |
Taselisib | MINK | 88.0 | 100 | nM |