Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib EGFR(L858R) 99.0 100
nM
Taselisib EGFR(L858R) 90.0 1000
nM
Taselisib EGFR(L858R,T790M) 69.0 100
nM
Taselisib EGFR(L858R,T790M) 98.0 1000
nM
Taselisib EGFR(L861Q) 95.0 100
nM
Taselisib EGFR(L861Q) 79.0 1000
nM
Taselisib EGFR(S752-I759del) 93.0 100
nM
Taselisib EGFR(S752-I759del) 99.0 1000
nM
Taselisib EGFR(T790M) 90.0 100
nM
Taselisib EGFR(T790M) 100.0 1000
nM
Taselisib EIF2AK1 96.0 100
nM
Taselisib EIF2AK1 100.0 1000
nM
Taselisib EPHA1 100.0 100
nM
Taselisib EPHA1 100.0 1000
nM
Taselisib EPHA2 80.0 100
nM
Taselisib EPHA2 100.0 1000
nM
Taselisib EPHA3 94.0 100
nM
Taselisib EPHA3 98.0 1000
nM
Taselisib EPHA4 94.0 100
nM
Taselisib EPHA4 95.0 1000
nM
Taselisib EPHA5 96.0 100
nM
Taselisib EPHA5 95.0 1000
nM
Taselisib EPHA6 95.0 100
nM
Taselisib EPHA6 92.0 1000
nM
Taselisib EPHA7 98.0 100
nM