Taselisib KINOMEscan - Dataset (ID:20264)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Taselisib | EGFR(L858R) | 99.0 | 100 | nM |
Taselisib | EGFR(L858R) | 90.0 | 1000 | nM |
Taselisib | EGFR(L858R,T790M) | 69.0 | 100 | nM |
Taselisib | EGFR(L858R,T790M) | 98.0 | 1000 | nM |
Taselisib | EGFR(L861Q) | 95.0 | 100 | nM |
Taselisib | EGFR(L861Q) | 79.0 | 1000 | nM |
Taselisib | EGFR(S752-I759del) | 93.0 | 100 | nM |
Taselisib | EGFR(S752-I759del) | 99.0 | 1000 | nM |
Taselisib | EGFR(T790M) | 90.0 | 100 | nM |
Taselisib | EGFR(T790M) | 100.0 | 1000 | nM |
Taselisib | EIF2AK1 | 96.0 | 100 | nM |
Taselisib | EIF2AK1 | 100.0 | 1000 | nM |
Taselisib | EPHA1 | 100.0 | 100 | nM |
Taselisib | EPHA1 | 100.0 | 1000 | nM |
Taselisib | EPHA2 | 80.0 | 100 | nM |
Taselisib | EPHA2 | 100.0 | 1000 | nM |
Taselisib | EPHA3 | 94.0 | 100 | nM |
Taselisib | EPHA3 | 98.0 | 1000 | nM |
Taselisib | EPHA4 | 94.0 | 100 | nM |
Taselisib | EPHA4 | 95.0 | 1000 | nM |
Taselisib | EPHA5 | 96.0 | 100 | nM |
Taselisib | EPHA5 | 95.0 | 1000 | nM |
Taselisib | EPHA6 | 95.0 | 100 | nM |
Taselisib | EPHA6 | 92.0 | 1000 | nM |
Taselisib | EPHA7 | 98.0 | 100 | nM |