Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib DMPK2 100.0 1000
nM
Taselisib DRAK1 100.0 100
nM
Taselisib DRAK1 97.0 1000
nM
Taselisib DRAK2 94.0 100
nM
Taselisib DRAK2 97.0 1000
nM
Taselisib DYRK1A 83.0 100
nM
Taselisib DYRK1A 99.0 1000
nM
Taselisib DYRK1B 74.0 100
nM
Taselisib DYRK1B 84.0 1000
nM
Taselisib DYRK2 93.0 100
nM
Taselisib DYRK2 64.0 1000
nM
Taselisib EGFR 96.0 100
nM
Taselisib EGFR 93.0 1000
nM
Taselisib EGFR(E746-A750del) 89.0 100
nM
Taselisib EGFR(E746-A750del) 97.0 1000
nM
Taselisib EGFR(G719C) 93.0 100
nM
Taselisib EGFR(G719C) 97.0 1000
nM
Taselisib EGFR(G719S) 98.0 100
nM
Taselisib EGFR(G719S) 86.0 1000
nM
Taselisib EGFR(L747-E749del, A750P) 100.0 100
nM
Taselisib EGFR(L747-E749del, A750P) 87.0 1000
nM
Taselisib EGFR(L747-S752del, P753S) 88.0 100
nM
Taselisib EGFR(L747-S752del, P753S) 91.0 1000
nM
Taselisib EGFR(L747-T751del,Sins) 88.0 100
nM
Taselisib EGFR(L747-T751del,Sins) 84.0 1000
nM