Taselisib KINOMEscan - Dataset (ID:20264)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Taselisib | RET(V804M) | 99.0 | 100 | nM |
Taselisib | RET(V804M) | 100.0 | 1000 | nM |
Taselisib | RIOK1 | 67.0 | 100 | nM |
Taselisib | RIOK1 | 75.0 | 1000 | nM |
Taselisib | RIOK2 | 91.0 | 100 | nM |
Taselisib | RIOK2 | 99.0 | 1000 | nM |
Taselisib | RIOK3 | 71.0 | 100 | nM |
Taselisib | RIOK3 | 95.0 | 1000 | nM |
Taselisib | RIPK1 | 98.0 | 100 | nM |
Taselisib | RIPK1 | 100.0 | 1000 | nM |
Taselisib | RIPK2 | 97.0 | 100 | nM |
Taselisib | RIPK2 | 85.0 | 1000 | nM |
Taselisib | RIPK4 | 100.0 | 100 | nM |
Taselisib | RIPK4 | 98.0 | 1000 | nM |
Taselisib | RIPK5 | 81.0 | 100 | nM |
Taselisib | RIPK5 | 99.0 | 1000 | nM |
Taselisib | ROCK1 | 100.0 | 100 | nM |
Taselisib | ROCK1 | 98.0 | 1000 | nM |
Taselisib | ROCK2 | 100.0 | 100 | nM |
Taselisib | ROCK2 | 91.0 | 1000 | nM |
Taselisib | ROS1 | 96.0 | 100 | nM |
Taselisib | ROS1 | 100.0 | 1000 | nM |
Taselisib | RPS6KA4(Kin.Dom.1-N-terminal) | 95.0 | 100 | nM |
Taselisib | RPS6KA4(Kin.Dom.1-N-terminal) | 88.0 | 1000 | nM |
Taselisib | RPS6KA4(Kin.Dom.2-C-terminal) | 88.0 | 100 | nM |