Taselisib KINOMEscan - Dataset (ID:20264)

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Small Molecule Protein % Control Assay compound conc Conc unit
Taselisib RET(V804M) 99.0 100
nM
Taselisib RET(V804M) 100.0 1000
nM
Taselisib RIOK1 67.0 100
nM
Taselisib RIOK1 75.0 1000
nM
Taselisib RIOK2 91.0 100
nM
Taselisib RIOK2 99.0 1000
nM
Taselisib RIOK3 71.0 100
nM
Taselisib RIOK3 95.0 1000
nM
Taselisib RIPK1 98.0 100
nM
Taselisib RIPK1 100.0 1000
nM
Taselisib RIPK2 97.0 100
nM
Taselisib RIPK2 85.0 1000
nM
Taselisib RIPK4 100.0 100
nM
Taselisib RIPK4 98.0 1000
nM
Taselisib RIPK5 81.0 100
nM
Taselisib RIPK5 99.0 1000
nM
Taselisib ROCK1 100.0 100
nM
Taselisib ROCK1 98.0 1000
nM
Taselisib ROCK2 100.0 100
nM
Taselisib ROCK2 91.0 1000
nM
Taselisib ROS1 96.0 100
nM
Taselisib ROS1 100.0 1000
nM
Taselisib RPS6KA4(Kin.Dom.1-N-terminal) 95.0 100
nM
Taselisib RPS6KA4(Kin.Dom.1-N-terminal) 88.0 1000
nM
Taselisib RPS6KA4(Kin.Dom.2-C-terminal) 88.0 100
nM