5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | MWCL.1 | AurB | SHFIVALKVLFK | Lys1 | -23.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | 31.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | -9.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | -1.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CAMK1D | LFAVKCIPK | Lys1 | 2.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | -3.8 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | KCC4 | DLKPENLLYATPAPDAPLK | Lys2 | 27.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CaMKK2 | DIKPSNLLVGEDGHIK | Lys2 | -16.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CASK | ETGQQFAVKIVDVAK | Lys1 | -22.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | -2.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | 37.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | -9.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | 9.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CDK5 | DLKPQNLLINR | Lys2 | -4.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | 1.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | -30.3 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CDK9 | DMKAANVLITR | Lys2 | 25.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CHK1 | DIKPENLLLDER | Lys2 | -21.7 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | -25.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CK1d,CK1e | DVKPDNFLMGLGKK | Lys2 | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | CK2a2 | DVKPHNVMIDHQQK | Lys2 | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | CLK3 | YEIVGNLGEGTFGKVVECLDHAR | ATP Loop | 2.2 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | -3.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | DGKA | IDPVPNTHPLLVFVNPKSGGK | ATP | -18.8 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | DNAPK | EHPFLVKGGEDLR | ATP | 41.3 | 1 | uM |