5z-7-oxozeaenol KiNativ -- single dose experiment - Dataset (ID:20255)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| 5z-7-oxozeaenol | BCWM.1 | MK11 | QELNKTVWEVPQR | Other | 5.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KS6B1 | DLKPENIMLNHQGHVK | Lys2 | -44.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | KS6B2 | DLKPENIMLSSQGHIK | Lys2 | 15.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CDK16 | SKLTDNLVALKEIR | Lys1 | -10.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | CDK14 | LVALKVIR | Lys1 | 7.5 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | 22.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | FAK2 | YIEDEDYYKASVTR | Activation Loop | 27.1 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | RSK1_domain2 | DLKPSNILYVDESGNPECLR | Lys2 | 16.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | RSK1,RSK2,RSK3_domain1 | DLKPENILLDEEGHIK | Lys2 | 13.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | RSK2_domain2 | DLKPSNILYVDESGNPESIR | Lys2 | 2.7 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | RSK3_domain1 | DLKPENILLDEEGHIKITDFGLSK | Lys2 | 8.2 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | RSKL1_domain1 | VLGVIDKVLLVMDTR | Protein Kinase Domain | 4.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | SRPK1/2 | FVAMKVVK | Lys1 | 5.9 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | MAP3K7,TAK1 | DLKPPNLLLVAGGTVLK | Lys2 | 97.0 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | Lys2 | 6.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TAOK2 | DVKAGNILLSEPGLVK | Lys2 | 14.8 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | 2.4 | 1 | uM |
| 5z-7-oxozeaenol | BCWM.1 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 11.1 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | 25.9 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 17.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | AGK | ATVFLNPAACKGK | Other | 1 | uM | |
| 5z-7-oxozeaenol | MWCL.1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 23.0 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | -120.6 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | ATR | FYIMMCKPK | ATP | 28.5 | 1 | uM |
| 5z-7-oxozeaenol | MWCL.1 | AurA | FILALKVLFK | Lys1 | -15.2 | 1 | uM |