PF-3758309 KiNativ -- single dose experiment - Dataset (ID:20254)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
PF-3758309 THP-1 PRPK
FLSGLELVKQGAEAR
ATP Loop
12.4
 1
uM
PF-3758309 THP-1 FAK2
YIEDEDYYKASVTR
Activation Loop
63.9
 1
uM
PF-3758309 THP-1 SIK3
VAIKIIDKTQLDEENLKK
Lys1
25.0
 1
uM
PF-3758309 THP-1 RIPK3
DLKPSNVLLDPELHVK
Lys2
-14.0
 1
uM
PF-3758309 THP-1 RSK1,RSK2,RSK3_domain1
DLKPENILLDEEGHIK
Lys2
90.6
 1
uM
PF-3758309 THP-1 RSK1 (Domain 2)
ATNMEYAVKVIDK
Lys1
-23.7
 1
uM
PF-3758309 THP-1 RSK2_domain2
DLKPSNILYVDESGNPESIR
Lys2
-6.9
 1
uM
PF-3758309 THP-1 SGK3
FYAVKVLQK
Lys1
-16.1
 1
uM
PF-3758309 THP-1 SLK
DLKAGNILFTLDGDIK
Lys2
17.6
 1
uM
PF-3758309 THP-1 SNRK
DLKPENVVFFEK
Lys2
-7.9
 1
uM
PF-3758309 THP-1 SRPK1/2
FVAMKVVK
Lys1
89.2
 1
uM
PF-3758309 THP-1 STLK6
HTPTGTLVTIKITNLENCNEER
Lys1
-12.8
 1
uM
PF-3758309 THP-1 SYK
TVAVKILK
Lys1
6.7
 1
uM
PF-3758309 THP-1 TLK2
YVAVKIHQLNK
Lys1
64.3
 1
uM
PF-3758309 THP-1 ULK1
DLKPQNILLSNPAGR
Lys2
-9.5
 1
uM
PF-3758309 THP-1 ULK3
EVVAIKCVAK
Lys1
41.4
 1
uM
PF-3758309 THP-1 Wnk1,Wnk2,Wnk3
DLKCDNIFITGPTGSVK
Lys2
0.9
 1
uM
PF-3758309 THP-1 Wnk1,Wnk2,Wnk4
IGDLGLATLKR
Activation Loop
-3.8
 1
uM
PF-3758309 THP-1 MLTK
WISQDKEVAVKK
Lys1
-6.3
 1
uM
PF-3758309 THP-1 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIKGQNVLLTENAEVK
Lys2
8.4
 1
uM
PF-3758309 THP-1 M4K3
NVNTGELAAIKVIK
Lys1
28.7
 1
uM
PF-3758309 THP-1 MARK3
EVAIKIIDKTQLNPTSLQK
Lys1
89.4
 1
uM
PF-3758309 THP-1 PIP4K2A
AKELPTLKDNDFINEGQK
ATP
4.1
 1
uM
PF-3758309 THP-1 MAP3K5,MAP3K6,MAP3K7
IAIKEIPERDSR
Lys1
-3.8
 1
uM