PF-3758309 KiNativ -- single dose experiment - Dataset (ID:20254)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
PF-3758309 THP-1 IRAK4
DIKSANILLDEAFTAK
Lys2
4.0
 1
uM
PF-3758309 THP-1 JNK1,JNK2,JNK3
DLKPSNIVVK
Lys2
1.0
 1
uM
PF-3758309 THP-1 KHS1
NVHTGELAAVKIIK
Lys1
22.1
 1
uM
PF-3758309 THP-1 LATS1
ALYATKTLR
Lys1
-51.4
 1
uM
PF-3758309 THP-1 LKB1
DIKPGNLLLTTGGTLK
Lys2
84.9
 1
uM
PF-3758309 THP-1 LOK
NKETGALAAAKVIETK
Lys1
23.7
 1
uM
PF-3758309 THP-1 MAP2K1,MAP2K2
DVKPSNILVNSR
Lys2
-6.6
 1
uM
PF-3758309 THP-1 MAP2K3
DVKPSNVLINK
Lys2
-7.5
 1
uM
PF-3758309 THP-1 MAP2K4
MVHKPSGQIMAVKR
Lys1
-10.8
 1
uM
PF-3758309 THP-1 MAP2K5
DVKPSNMLVNTR
Lys2
-18.2
 1
uM
PF-3758309 THP-1 MAP2K6
HVPSGQIMAVKR
Lys1
-16.4
 1
uM
PF-3758309 THP-1 MAP2K6
DVKPSNVLINALGQVK
Lys2
21.2
 1
uM
PF-3758309 THP-1 MP2K7
DVKPSNILLDER
Lys2
14.7
 1
uM
PF-3758309 THP-1 MAP3K1
DVKGANLLIDSTGQR
Lys2
-9.4
 1
uM
PF-3758309 THP-1 M3K2,MAP3K3
DIKGANILR
Lys2
10.7
 1
uM
PF-3758309 THP-1 MARK1,MARK2
EVAVKIIDK
Lys1
90.2
 1
uM
PF-3758309 THP-1 MARK3,MARK4
EVAIKIIDK
Lys1
90.1
 1
uM
PF-3758309 THP-1 MASTL
LYAVKVVK
Lys1
-8.2
 1
uM
PF-3758309 THP-1 MER,TYRO3
KIYSGDYYR
Activation Loop
74.2
 1
uM
PF-3758309 THP-1 MLK3
DLKSNNILLLQPIESDDMEHK
Lys2
45.0
 1
uM
PF-3758309 THP-1 MST1
ETGQIVAIKQVPVESDLQEIIK
Lys1
74.3
 1
uM
PF-3758309 THP-1 MST1,MST2
DIKAGNILLNTEGHAK
Lys2
43.9
 1
uM
PF-3758309 THP-1 MST2
ESGQVVAIKQVPVESDLQEIIK
Lys1
73.0
 1
uM
PF-3758309 THP-1 MST4,YSK1
DIKAANVLLSEQGDVK
Lys2
76.4
 1
uM
PF-3758309 THP-1 NDR1
DTGHVYAMKILR
Lys1
47.1
 1
uM