PF-3758309 KiNativ -- single dose experiment - Dataset (ID:20254)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| PF-3758309 | THP-1 | NEK7 | AACLLDGVPVALKK | Lys1 | -13.2 | 1 | uM |
| PF-3758309 | THP-1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 8.6 | 1 | uM |
| PF-3758309 | THP-1 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | 4.1 | 1 | uM |
| PF-3758309 | THP-1 | LATS1 | ALYATKTLR | Lys1 | -51.4 | 1 | uM |
| PF-3758309 | THP-1 | RSK1 (Domain 2) | ATNMEYAVKVIDK | Lys1 | -23.7 | 1 | uM |
| PF-3758309 | THP-1 | PLK1 | CFEISDADTKEVFAGKIVPK | Lys1 | 2.5 | 1 | uM |
| PF-3758309 | THP-1 | FAK | CIGEGQFGDVHQGIYMSPENPALAVAIKTCK | Lys1 | 23.2 | 1 | uM |
| PF-3758309 | THP-1 | MST4,YSK1 | DIKAANVLLSEQGDVK | Lys2 | 76.4 | 1 | uM |
| PF-3758309 | THP-1 | MST1,MST2 | DIKAGNILLNTEGHAK | Lys2 | 43.9 | 1 | uM |
| PF-3758309 | THP-1 | CDK13 | DIKCSNILLNNR | Lys2 | -7.4 | 1 | uM |
| PF-3758309 | THP-1 | CRK7 | DIKCSNILLNNSGQIK | Lys2 | 8.2 | 1 | uM |
| PF-3758309 | THP-1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | 10.7 | 1 | uM |
| PF-3758309 | THP-1 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | 8.4 | 1 | uM |
| PF-3758309 | THP-1 | NEK6,NEK7 | DIKPANVFITATGVVK | Lys2 | -4.4 | 1 | uM |
| PF-3758309 | THP-1 | IKKE,TBK1 | DIKPGNIMR | Lys2 | 87.6 | 1 | uM |
| PF-3758309 | THP-1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 84.9 | 1 | uM |
| PF-3758309 | THP-1 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | 74.7 | 1 | uM |
| PF-3758309 | THP-1 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | 52.6 | 1 | uM |
| PF-3758309 | THP-1 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | 4.0 | 1 | uM |
| PF-3758309 | THP-1 | NEK1 | DIKSQNIFLTK | Lys2 | 7.3 | 1 | uM |
| PF-3758309 | THP-1 | NEK9 | DIKTLNIFLTK | Lys2 | 36.6 | 1 | uM |
| PF-3758309 | THP-1 | HPK1 | DKVSGDLVALKMVK | Lys1 | 15.1 | 1 | uM |
| PF-3758309 | THP-1 | SLK | DLKAGNILFTLDGDIK | Lys2 | 17.6 | 1 | uM |
| PF-3758309 | THP-1 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | 0.9 | 1 | uM |
| PF-3758309 | THP-1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | -29.4 | 1 | uM |