LINCS Pilot Phase Joint Project: Sensitivity measures of six breast cancer cell lines to a library of small molecule kinase inhibitors (single drug treatments). Dataset 5 of 15: Mean cell count and mean growth rate across biological replicate 2. - Dataset (ID:20241)
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Cell | Small Molecule | Small Mol Concentration | Small Mol Conc Unit | LJP Library Plate | Timepoint | Timepoint Unit | Mean Total Cell Count Before Treatment | Mean Total Cell Count After Treatment | Mean Total Control Cell Count | Mean Relative Cell Count | Mean Relative Growth Rate After Treatment |
---|---|---|---|---|---|---|---|---|---|---|---|
Hs 578T | WZ3105 | 10.0 | uM | LJP5 | 72 | hr | 765 | 386 | 3124 | 0.1236 | -0.1605 |
Hs 578T | XMD11-50 | 10.0 | uM | LJP6 | 72 | hr | 765 | 548 | 3124 | 0.1756 | -0.0917 |
Hs 578T | Y39983 | 10.0 | uM | LJP6 | 72 | hr | 765 | 740 | 3124 | 0.2369 | -0.0105 |
Hs 578T | YM 201636 | 10.0 | uM | LJP5 | 72 | hr | 765 | 955 | 3124 | 0.3059 | 0.0808 |
Hs 578T | ZSTK474 | 10.0 | uM | LJP6 | 72 | hr | 765 | 805 | 3124 | 0.2579 | 0.0172 |
MCF 10A | Afatinib | 0.04 | uM | LJP6 | 72 | hr | 1694 | 1726 | 11155 | 0.1548 | 0.0034 |
MCF 10A | Sigma A6730 | 0.04 | uM | LJP5 | 72 | hr | 1694 | 11014 | 11155 | 0.9874 | 0.9851 |
MCF 10A | Alvocidib | 0.04 | uM | LJP6 | 72 | hr | 1694 | 4715 | 11155 | 0.4227 | 0.3193 |
MCF 10A | AT-7519 | 0.04 | uM | LJP6 | 72 | hr | 1694 | 11122 | 11155 | 0.9970 | 0.9965 |
MCF 10A | AZD 5438 | 0.04 | uM | LJP6 | 72 | hr | 1694 | 10915 | 11155 | 0.9784 | 0.9746 |
MCF 10A | AZD-6482 | 0.04 | uM | LJP5 | 72 | hr | 1694 | 11212 | 11155 | 1.0051 | 1.0060 |
MCF 10A | AZD7762 | 0.04 | uM | LJP6 | 72 | hr | 1694 | 9157 | 11155 | 0.8208 | 0.7888 |
MCF 10A | AZD8055 | 0.04 | uM | LJP6 | 72 | hr | 1694 | 6286 | 11155 | 0.5635 | 0.4853 |
MCF 10A | AZD8330 | 0.04 | uM | LJP5 | 72 | hr | 1694 | 2625 | 11155 | 0.2353 | 0.0984 |
MCF 10A | Barasertib | 0.04 | uM | LJP5 | 72 | hr | 1694 | 2690 | 11155 | 0.2412 | 0.1053 |
MCF 10A | BI-2536 | 0.04 | uM | LJP6 | 72 | hr | 1694 | 1015 | 11155 | 0.0910 | -0.0717 |
MCF 10A | BMS345541 | 0.04 | uM | LJP6 | 72 | hr | 1694 | 11087 | 11155 | 0.9939 | 0.9928 |
MCF 10A | SNS-032 | 0.04 | uM | LJP6 | 72 | hr | 1694 | 11126 | 11155 | 0.9973 | 0.9969 |
MCF 10A | GDC-0980 | 0.04 | uM | LJP5 | 72 | hr | 1694 | 10202 | 11155 | 0.9145 | 0.8992 |
MCF 10A | NVP-AEW541 | 0.04 | uM | LJP5 | 72 | hr | 1694 | 10983 | 11155 | 0.9846 | 0.9818 |
MCF 10A | SB590885 | 0.04 | uM | LJP5 | 72 | hr | 1694 | 11109 | 11155 | 0.9959 | 0.9951 |
MCF 10A | PIK-93 | 0.04 | uM | LJP5 | 72 | hr | 1694 | 11144 | 11155 | 0.9990 | 0.9988 |
MCF 10A | KIN001-043 | 0.04 | uM | LJP6 | 72 | hr | 1694 | 11293 | 11155 | 1.0123 | 1.0146 |
MCF 10A | Alpelisib | 0.04 | uM | LJP5 | 72 | hr | 1694 | 10662 | 11155 | 0.9558 | 0.9479 |
MCF 10A | Luminespib | 0.04 | uM | LJP5 | 72 | hr | 1694 | 1257 | 11155 | 0.1127 | -0.0462 |