JNK-IN-8 KiNativ -- single dose experiment - Dataset (ID:20213)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| JNK-IN-8 | A-375 | NEK7 | FFSSkTTAAHSLVGTPYYMSPER | Activation Loop | -1.1 | 1 | uM |
| JNK-IN-8 | A-375 | NEK7 | AACLLDGVPVALkK | Lys1 | -26.5 | 1 | uM |
| JNK-IN-8 | A-375 | NEK8 | DLkTQNILLDK | Lys2 | -9.6 | 1 | uM |
| JNK-IN-8 | A-375 | NEK9 | LGDYGLAkK | Activation Loop | 12.1 | 1 | uM |
| JNK-IN-8 | A-375 | NEK9 | RTEDDSLVVWkEVDLTR | Lys1 | -29.4 | 1 | uM |
| JNK-IN-8 | A-375 | NEK9 | DIkTLNIFLTK | Lys2 | -32.2 | 1 | uM |
| JNK-IN-8 | A-375 | OSR1 | DVkAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | -4.0 | 1 | uM |
| JNK-IN-8 | A-375 | OSR1 | NGQIHRDVkAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | 5.1 | 1 | uM |
| JNK-IN-8 | A-375 | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | -8.9 | 1 | uM |
| JNK-IN-8 | A-375 | KS6B1 | LTDFGLCkESIHDGTVTHTFCGTIEYMAPEILMR | Activation Loop | -0.6 | 1 | uM |
| JNK-IN-8 | A-375 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | -37.6 | 1 | uM |
| JNK-IN-8 | A-375 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | -26.5 | 1 | uM |
| JNK-IN-8 | A-375 | KS6B2 | LTDFGLCkESIHEGAVTHTFCGTIEYMAPEILVR | Activation Loop | 33.1 | 1 | uM |
| JNK-IN-8 | A-375 | KS6B2 | DLkPENIMLSSQGHIK | Lys2 | -29.1 | 1 | uM |
| JNK-IN-8 | A-375 | CDK16 | LTDNLVALkEIR | Lys1 | -9.0 | 1 | uM |
| JNK-IN-8 | A-375 | PCTAIRE2 | DLkPQNLLINEK | Lys2 | 16.5 | 1 | uM |
| JNK-IN-8 | A-375 | PCTAIRE2,PCTAIRE3 | SKLTENLVALkEIRLEHEEGAPCTAIR | Lys1 | 13.0 | 1 | uM |
| JNK-IN-8 | A-375 | PCTAIRE2,PCTAIRE3 | SKLTENLVALkEIR | Lys1 | 4.4 | 1 | uM |
| JNK-IN-8 | A-375 | PDK1 | HIIKENkVPYVTR | Protein Kinase Domain | -10.9 | 1 | uM |
| JNK-IN-8 | A-375 | CDK14 | LVALkVIR | Lys1 | 38.1 | 1 | uM |
| JNK-IN-8 | A-375 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | -0.8 | 1 | uM |
| JNK-IN-8 | A-375 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 12.3 | 1 | uM |
| JNK-IN-8 | A-375 | PI4KB | VPHTQAVVLNSkDK | ATP | 8.0 | 1 | uM |
| JNK-IN-8 | A-375 | PI4KB | VPHTQAVVLNSKDkAPYLIYVEVLECENFDTTSVPAR | ATP | 25.0 | 1 | uM |
| JNK-IN-8 | A-375 | PIK3C3 | TEDGGKYPVIFkHGDDLRQDQLILQIISLMDK | ATP | 18.1 | 1 | uM |