JNK-IN-8 KiNativ -- single dose experiment - Dataset (ID:20213)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JNK-IN-8 A-375 WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
-68.7
1
uM
JNK-IN-8 A-375 Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
12.7
1
uM
JNK-IN-8 A-375 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-15.1
1
uM
JNK-IN-8 A-375 WNK4
DLkCDNVFITGPTGSVK
Lys2
16.1
1
uM
JNK-IN-8 A-375 MLTK
WISQDKEVAVKk
Lys1
-7.8
1
uM
JNK-IN-8 A-375 ZC1/HGK
TGQLAAIkVMDVTEDEEEEIKLEINMLK
Lys1
44.8
1
uM
JNK-IN-8 A-375 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-11.3
1
uM
JNK-IN-8 A-375 ZC2/TNIK
TGQLAAIkVMDVTGDEEEEIKQEINMLKK
Lys1
9.9
1
uM
JNK-IN-8 A-375 ZC2/TNIK,ZC3/MINK
VIHRDIkGQNVLLTENAEVK
Lys2
45.1
1
uM
JNK-IN-8 A-375 MK14
QELNkTIWEVPER
Other
3.9
1
uM
JNK-IN-8 A-375 PAN3
VMDPTkILITGK
Protein Kinase Domain
-34.7
1
uM
JNK-IN-8 A-375 PIK4CB
VPHTQAVVLNSkDKAPYLIYVEVLECENFDTTSVPARIPENR
ATP
10.1
1
uM
JNK-IN-8 A-375 PIK3CD
TkVNWLAHNVSKDNRQ
ATP
22.9
1
uM
JNK-IN-8 A-375 PRKACB
DLkPENLLIDHQGYIQ
Lys2
12.8
1
uM
JNK-IN-8 A-375 p38a
DLkPSNLAVNEDCELK
Lys2
13.2
1
uM