JNK-IN-8 KiNativ -- single dose experiment - Dataset (ID:20213)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| JNK-IN-8 | A-375 | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | -28.5 | 1 | uM |
| JNK-IN-8 | A-375 | MLKL | APVAIkVFK | Lys1 | 11.6 | 1 | uM |
| JNK-IN-8 | A-375 | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | -30.3 | 1 | uM |
| JNK-IN-8 | A-375 | MSK1_domain1 | DIkLENILLDSNGHVVLTDFGLSK | Lys2 | -3.1 | 1 | uM |
| JNK-IN-8 | A-375 | MST1 | AIHKETGQIVAIkQVPVESDLQEIIK | Lys1 | -2.6 | 1 | uM |
| JNK-IN-8 | A-375 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 0.5 | 1 | uM |
| JNK-IN-8 | A-375 | MST1,MST2 | IHRDIkAGNILLNTEGHAK | Lys2 | -10.9 | 1 | uM |
| JNK-IN-8 | A-375 | MST1,MST2 | DIkAGNILLNTEGHAK | Lys2 | -3.9 | 1 | uM |
| JNK-IN-8 | A-375 | MST2 | ESGQVVAIkQVPVESDLQEIIK | Lys1 | 10.0 | 1 | uM |
| JNK-IN-8 | A-375 | MST2 | ESGQVVAIkQVPVESDLQEIIKEISIMQQCDSPYVVK | Lys1 | 25.6 | 1 | uM |
| JNK-IN-8 | A-375 | MST3 | DIkAANVLLSEHGEVK | Lys2 | -0.9 | 1 | uM |
| JNK-IN-8 | A-375 | MST3 | IHRDIkAANVLLSEHGEVK | Lys2 | -24.0 | 1 | uM |
| JNK-IN-8 | A-375 | MST3,MST4,YSK1 | LADFGVAGQLTDTQIkR | Activation Loop | 19.4 | 1 | uM |
| JNK-IN-8 | A-375 | MST4,YSK1 | IHRDIkAANVLLSEQGDVK | Lys2 | 15.3 | 1 | uM |
| JNK-IN-8 | A-375 | MST4,YSK1 | DIkAANVLLSEQGDVK | Lys2 | -2.2 | 1 | uM |
| JNK-IN-8 | A-375 | NDR1 | KDTGHVYAMkILR | Lys1 | -22.7 | 1 | uM |
| JNK-IN-8 | A-375 | NDR1 | DTGHVYAMkILR | Lys1 | -10.9 | 1 | uM |
| JNK-IN-8 | A-375 | NDR1 | DIkPDNLLLDSK | Lys2 | 5.8 | 1 | uM |
| JNK-IN-8 | A-375 | NDR1,NDR2 | LSDFGLCTGLkK | Activation Loop | -6.6 | 1 | uM |
| JNK-IN-8 | A-375 | NDR2 | KDTGHIYAMkILR | Lys1 | -20.1 | 1 | uM |
| JNK-IN-8 | A-375 | NDR2 | DTGHIYAMkILR | Lys1 | -29.0 | 1 | uM |
| JNK-IN-8 | A-375 | NDR2 | DIkPDNLLLDAK | Lys2 | 14.7 | 1 | uM |
| JNK-IN-8 | A-375 | NEK1 | DIkSQNIFLTK | Lys2 | -12.1 | 1 | uM |
| JNK-IN-8 | A-375 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -10.2 | 1 | uM |
| JNK-IN-8 | A-375 | NEK6,NEK7 | VMHRDIkPANVFITATGVVK | Lys2 | 15.5 | 1 | uM |