OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| OTSSP167 | MDA-MB-468 | FRK | HEIKLPVK | Activation Loop | 87.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | GPRK5 | DLKPENILLDDYGHIR | Lys2 | 88.2 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ERBB3 | GVWIPEGESIKIPVCIKVIEDK | Lys1 | 47.1 | 1 | uM |
| OTSSP167 | MDA-MB-468 | MK09 | YQQLKPIGSGAQGIVCAAFDTVLGINVAVKK | Lys1 | 44.1 | 1 | uM |
| OTSSP167 | MDA-MB-468 | MARK4 | DLKAENLLLDAEANIK | Lys2 | >97 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PKMYT1 | DTLLALAHLHSQGLVHLDVKPANIFLGPR | Lys2 | 65.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | NEK2 | DLKPANVFLDGK | Lys2 | 61.1 | 1 | uM |
| OTSSP167 | MDA-MB-468 | NUAK1 | LVAIKSIR | Lys1 | >96 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 88.4 | 1 | uM |
| OTSSP167 | MDA-MB-468 | YES | VAIKTLKPGTMMPEAFLQEAQIMK | Lys1 | >88 | 1 | uM |
| OTSSP167 | MDA-MB-468 | KCC4 | DLKPENLLYATPAPDAPLK | Lys2 | 93.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDK13 | DIKCSNILLNNR | Lys2 | 56.1 | 1 | uM |
| OTSSP167 | MDA-MB-468 | EPHB3 | FLEDDPSDPTYTSSLGGKIPIR | Activation Loop | 93.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 1.5 | 1 | uM |
| OTSSP167 | MDA-MB-468 | M3K6 | DIKGDNVLINTFSGLLK | Lys2 | 38.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | P4K2B | SEEPYGQLNPKWTK | ATP | 4.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | RSK2 domain1 | DLKPENILLDEEGHIKLTDFGLSKESIDHEK | Lys2 | >97 | 1 | uM |
| OTSSP167 | MDA-MB-468 | SGK1 | HKAEEVFYAVKVLQK | Lys1 | >98 | 1 | uM |