OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
OTSSP167 | MDA-MB-468 | RSK2_domain2 | DLKPSNILYVDESGNPESIR | Lys2 | >97 | 1 | uM |
OTSSP167 | MDA-MB-468 | RSKL1_domain1 | VLGVIDKVLLVMDTR | ATP | -41.3 | 1 | uM |
OTSSP167 | MDA-MB-468 | SGK3 | FYAVKVLQK | Lys1 | 91.5 | 1 | uM |
OTSSP167 | MDA-MB-468 | SLK | DLKAGNILFTLDGDIK | Lys2 | 93.4 | 1 | uM |
OTSSP167 | MDA-MB-468 | SMG1 | DTVTIHSVGGTITILPTKTKPK | ATP | 98.1 | 1 | uM |
OTSSP167 | MDA-MB-468 | SNRK | DLKPENVVFFEK | Lys2 | 12.8 | 1 | uM |
OTSSP167 | MDA-MB-468 | SRPK1 | IIHTDIKPENILLSVNEQYIR | Lys2 | 86.8 | 1 | uM |
OTSSP167 | MDA-MB-468 | SRPK1/2 | FVAMKVVK | Lys1 | 72.8 | 1 | uM |
OTSSP167 | MDA-MB-468 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | 83.5 | 1 | uM |
OTSSP167 | MDA-MB-468 | SYK | ISDFGLSKALR | Activation Loop | 91.6 | 1 | uM |
OTSSP167 | MDA-MB-468 | MAP3K7,TAK1 | DLKPPNLLLVAGGTVLK | Lys2 | >93 | 1 | uM |
OTSSP167 | MDA-MB-468 | TAO1,TAOK3 | DIKAGNILLTEPGQVK | Lys2 | >99 | 1 | uM |
OTSSP167 | MDA-MB-468 | TAOK2 | DVKAGNILLSEPGLVK | Lys2 | >97 | 1 | uM |
OTSSP167 | MDA-MB-468 | TBK1 | TGDLFAIKVFNNISFLRPVDVQMR | Lys1 | >90 | 1 | uM |
OTSSP167 | MDA-MB-468 | TLK1 | YLNEIKPPIIHYDLKPGNILLVDGTACGEIK | Lys2 | 53.7 | 1 | uM |
OTSSP167 | MDA-MB-468 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | 16.7 | 1 | uM |
OTSSP167 | MDA-MB-468 | TNK1 | SVPVAVKSLR | Lys1 | >95 | 1 | uM |
OTSSP167 | MDA-MB-468 | ULK1 | DLKPQNILLSNPAGR | Lys2 | -64.2 | 1 | uM |
OTSSP167 | MDA-MB-468 | ULK3 | NISHLDLKPQNILLSSLEKPHLK | Lys2 | 75.3 | 1 | uM |
OTSSP167 | MDA-MB-468 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | 12.6 | 1 | uM |
OTSSP167 | MDA-MB-468 | MLTK | WISQDKEVAVKK | Lys1 | >98 | 1 | uM |
OTSSP167 | MDA-MB-468 | ZC1/HGK,ZC2/TNIK,ZC3/MINK | DIKGQNVLLTENAEVK | Lys2 | >98 | 1 | uM |
OTSSP167 | MDA-MB-468 | KCC2D | IPTGQEYAAKIINTKK | Lys1 | 93.1 | 1 | uM |
OTSSP167 | MDA-MB-468 | CDK20 | DLKPANLLISASGQLK | Lys2 | 81.5 | 1 | uM |
OTSSP167 | MDA-MB-468 | KC1G2 | DVKPENFLVGRPGTK | Lys2 | 89.7 | 1 | uM |