OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| OTSSP167 | MDA-MB-468 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | 95.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ACK | TVSVAVKCLKPDVLSQPEAMDDFIR | Lys1 | 72.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 98.2 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ATR | FYIMMCKPK | ATP | >98 | 1 | uM |
| OTSSP167 | MDA-MB-468 | AurA | FILALKVLFK | Lys1 | 96.9 | 1 | uM |
| OTSSP167 | MDA-MB-468 | AurB | SHFIVALKVLFK | Lys1 | >99 | 1 | uM |
| OTSSP167 | MDA-MB-468 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | 7.6 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CaMK1a | LVAIKCIAK | Lys1 | 94.5 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CAMK1D | LFAVKCIPK | Lys1 | 75.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CaMK2g | TSTQEYAAKIINTK | Lys1 | 87.9 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CASK | ETGQQFAVKIVDVAK | Lys1 | 82.6 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | 96.9 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | 90.2 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | 98.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDK5 | DLKPQNLLINR | Lys2 | 94.6 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 95.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDK9 | DMKAANVLITR | Lys2 | 97.9 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CHK1 | DIKPENLLLDER | Lys2 | 94.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | >95 | 1 | uM |
| OTSSP167 | MDA-MB-468 | KC1A | DIKPDNFLMGIGR | Lys2 | 81.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CK1d,CK1e | DVKPDNFLMGLGKK | Lys2 | 85.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CLK2 | LTHTDLKPENILFVNSDYELTYNLEK | Lys2 | >95 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CLK3 | YEIVGNLGEGTFGKVVECLDHAR | ATP Loop | 98.4 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CRK7 | DIKCSNILLNNSGQIK | Lys2 | 59.6 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 92.1 | 1 | uM |