OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| OTSSP167 | MDA-MB-468 | IKKB | DLKPENIVLQQGEQR | Lys2 | -12.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | Wnk1,Wnk2,Wnk3 | DLKCDNIFITGPTGSVK | Lys2 | 12.6 | 1 | uM |
| OTSSP167 | MDA-MB-468 | NEK7 | AACLLDGVPVALKK | Lys1 | -12.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | SNRK | DLKPENVVFFEK | Lys2 | 12.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | MK03 | DLKPSNLLINTTCDLK | Lys2 | 1.5 | 1 | uM |
| OTSSP167 | MDA-MB-468 | MK01 | DLKPSNLLLNTTCDLK | Lys2 | 1.5 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TLK1/2 | YLNEIKPPIIHYDLKPGNILLVNGTACGEIK | Lys2 | 16.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ILK | WQGNDIVVKVLK | Lys1 | 18.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PAN3 | VMDPTKILITGK | ATP | -21.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | NEK3 | SKNIFLTQNGK | Activation Loop | 22.4 | 1 | uM |
| OTSSP167 | MDA-MB-468 | eEF2K | YIKYNSNSGFVR | ATP | -2.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | NEK6,NEK7 | DIKPANVFITATGVVK | Lys2 | 24.5 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ITPK1 | ESIFFNSHNVSKPESSSVLTELDKIEGVFERPSDEVIR | ATP | 25.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PKR | DLKPSNIFLVDTK | Lys2 | 25.9 | 1 | uM |
| OTSSP167 | MDA-MB-468 | MAP3K4 | DIKGANIFLTSSGLIK | Lys2 | 26.4 | 1 | uM |
| OTSSP167 | MDA-MB-468 | EGFR | LLGAEEKEYHAEGGKVPIK | Activation Loop | 29.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | M3K6 | DIKGDNVLINTFSGLLK | Lys2 | 38.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | RSKL1_domain1 | VLGVIDKVLLVMDTR | ATP | -41.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | JAK1 | QLASALSYLEDKDLVHGNVCTKNLLLAR | Protein Kinase Domain | 41.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | NEK8 | DLKTQNILLDK | Lys2 | 42.2 | 1 | uM |
| OTSSP167 | MDA-MB-468 | MK09 | YQQLKPIGSGAQGIVCAAFDTVLGINVAVKK | Lys1 | 44.1 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ERBB3 | GVWIPEGESIKIPVCIKVIEDK | Lys1 | 47.1 | 1 | uM |
| OTSSP167 | MDA-MB-468 | NEK1 | DIKSQNIFLTK | Lys2 | 47.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | P4K2B | SEEPYGQLNPKWTK | ATP | 4.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PIP4K2A | AKELPTLKDNDFINEGQK | ATP | 48.7 | 1 | uM |