OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| OTSSP167 | MDA-MB-468 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 92.1 | 1 | uM |
| OTSSP167 | MDA-MB-468 | STLK5 | YSVKVLPWLSPEVLQQNLQGYDAK | Activation Loop | 83.5 | 1 | uM |
| OTSSP167 | MDA-MB-468 | TYK2(Kin.Dom.2) | IGDFGLAKAVPEGHEYYR | Activation Loop | 88.4 | 1 | uM |
| OTSSP167 | MDA-MB-468 | EPHB4 | FLEENSSDPTYTSSLGGKIPIR | Activation Loop | >95 | 1 | uM |
| OTSSP167 | MDA-MB-468 | EGFR | LLGAEEKEYHAEGGKVPIK | Activation Loop | 29.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | SYK | ISDFGLSKALR | Activation Loop | 91.6 | 1 | uM |
| OTSSP167 | MDA-MB-468 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | 95.8 | 1 | uM |
| OTSSP167 | MDA-MB-468 | FRK | HEIKLPVK | Activation Loop | 87.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | MET | DMYDKEYYSVHNK | Activation Loop | >96 | 1 | uM |
| OTSSP167 | MDA-MB-468 | EPHB3 | FLEDDPSDPTYTSSLGGKIPIR | Activation Loop | 93.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | EphA1 | LLDDFDGTYETQGGKIPIR | Activation Loop | >97 | 1 | uM |
| OTSSP167 | MDA-MB-468 | NEK3 | SKNIFLTQNGK | Activation Loop | 22.4 | 1 | uM |
| OTSSP167 | MDA-MB-468 | EPHA2 | VLEDDPEATYTTSGGKIPIR | Activation Loop | >98 | 1 | uM |
| OTSSP167 | MDA-MB-468 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | 83.9 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | 95.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | >96 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PI4KA,PI4KAP2 | SGTPMQSAAKAPYLAK | ATP | 90.5 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PI4KB | VPHTQAVVLNSKDK | ATP | >98 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PAN3 | VMDPTKILITGK | ATP | -21.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PIK3C3 | TEDGGKYPVIFKHGDDLR | ATP | 90.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | PI42C | TLVIKEVSSEDIADMHSNLSNYHQYIVK | ATP | >97 | 1 | uM |
| OTSSP167 | MDA-MB-468 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | 92.1 | 1 | uM |
| OTSSP167 | MDA-MB-468 | ATR | FYIMMCKPK | ATP | >98 | 1 | uM |
| OTSSP167 | MDA-MB-468 | DNAPK | KGGSWIQEINVAEK | ATP | >97 | 1 | uM |
| OTSSP167 | MDA-MB-468 | DNAPK | EHPFLVKGGEDLR | ATP | 98.8 | 1 | uM |