OTSSP167 KiNativ -- single dose experiment - Dataset (ID:20209)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| OTSSP167 | MDA-MB-468 | PHKg1 | DLKPENILLDDNMNIK | Protein Kinase Domain | 92.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | JAK1 | QLASALSYLEDKDLVHGNVCTKNLLLAR | Protein Kinase Domain | 41.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | IRE1 | DLKPHNILISMPNAHGK | Lys2 | 68.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | IKKB | DLKPENIVLQQGEQR | Lys2 | -12.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | 97.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | 7.6 | 1 | uM |
| OTSSP167 | MDA-MB-468 | GCN2_domain2 | DLKPVNIFLDSDDHVK | Lys2 | 90.9 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDK9 | DMKAANVLITR | Lys2 | 97.9 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | 90.2 | 1 | uM |
| OTSSP167 | MDA-MB-468 | IKKA | DLKPENIVLQDVGGK | Lys2 | 5.2 | 1 | uM |
| OTSSP167 | MDA-MB-468 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 98.2 | 1 | uM |
| OTSSP167 | MDA-MB-468 | MK03 | DLKPSNLLINTTCDLK | Lys2 | 1.5 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | 98.7 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDK5 | DLKPQNLLINR | Lys2 | 94.6 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | 95.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | GCK | DIKGANLLLTLQGDVK | Lys2 | 96.5 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CHK1 | DIKPENLLLDER | Lys2 | 94.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | >95 | 1 | uM |
| OTSSP167 | MDA-MB-468 | KC1A | DIKPDNFLMGIGR | Lys2 | 81.0 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CK1d,CK1e | DVKPDNFLMGLGKK | Lys2 | 85.3 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CLK2 | LTHTDLKPENILFVNSDYELTYNLEK | Lys2 | >95 | 1 | uM |
| OTSSP167 | MDA-MB-468 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | >99 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CRK7 | DIKCSNILLNNSGQIK | Lys2 | 59.6 | 1 | uM |
| OTSSP167 | MDA-MB-468 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | >99 | 1 | uM |
| OTSSP167 | MDA-MB-468 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | 96.9 | 1 | uM |