QL-X-138 KiNativ -- single dose experiment - Dataset (ID:20204)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-X-138 | BCWM.1 | CSK | VSDFGLTKEASSTQDTGKLPVK | Activation Loop | 7.682513184 | 1 | uM |
| QL-X-138 | BCWM.1 | DNAPK | EHPFLVKGGEDLR | ATP | 41.71428541 | 1 | uM |
| QL-X-138 | BCWM.1 | DNAPK | KGGSWIQEINVAEK | ATP | 84.93363802 | 1 | uM |
| QL-X-138 | BCWM.1 | eEF2K | YIKYNSNSGFVR | ATP | -21.72541845 | 1 | uM |
| QL-X-138 | BCWM.1 | EPHB2 | FLEDDTSDPTYTSALGGKIPIR | Activation Loop | 82.85022013 | 1 | uM |
| QL-X-138 | BCWM.1 | MK03 | DLKPSNLLINTTCDLK | Lys2 | 8.257189818 | 1 | uM |
| QL-X-138 | BCWM.1 | FER | TSVAVKTCKEDLPQELK | Lys1 | 17.35545574 | 1 | uM |
| QL-X-138 | BCWM.1 | FES | LRADNTLVAVKSCR | Lys1 | 18.79754204 | 1 | uM |
| QL-X-138 | BCWM.1 | FGR | LIKDDEYNPCQGSKFPIK | Activation Loop | -1.765630814 | 1 | uM |
| QL-X-138 | BCWM.1 | FRAP1 | IQSIAPSLQVITSKQRPR | ATP | 80.6131392 | 1 | uM |
| QL-X-138 | BCWM.1 | FYN,SRC,YES | QGAKFPIKWTAPEAALYGR | Activation Loop | 62.9318999 | 1 | uM |
| QL-X-138 | BCWM.1 | GCK | DIKGANLLLTLQGDVK | Lys2 | -52.47193008 | 1 | uM |
| QL-X-138 | BCWM.1 | GCN2_domain2 | DLKPVNIFLDSDDHVK | Lys2 | 45.91026666 | 1 | uM |
| QL-X-138 | BCWM.1 | GSK3A | DIKPQNLLVDPDTAVLK | Lys2 | 12.82982094 | 1 | uM |
| QL-X-138 | BCWM.1 | GSK3B | DIKPQNLLLDPDTAVLK | Lys2 | -63.22002885 | 1 | uM |
| QL-X-138 | BCWM.1 | HPK1 | DIKGANILINDAGEVR | Lys2 | -3.2162289 | 1 | uM |
| QL-X-138 | BCWM.1 | IKKA | DLKPENIVLQDVGGK | Lys2 | 10.25359992 | 1 | uM |
| QL-X-138 | BCWM.1 | IKKB | DLKPENIVLQQGEQR | Lys2 | 21.13647451 | 1 | uM |
| QL-X-138 | BCWM.1 | IKKE | SGELVAVKVFNTTSYLRPR | Lys1 | 43.02362934 | 1 | uM |
| QL-X-138 | BCWM.1 | ILK | WQGNDIVVKVLK | Lys1 | 13.05452604 | 1 | uM |
| QL-X-138 | BCWM.1 | IRAK1 | AIQFLHQDSPSLIHGDIKSSNVLLDER | Lys2 | 70.76822338 | 1 | uM |
| QL-X-138 | BCWM.1 | IRAK4 | DIKSANILLDEAFTAK | Lys2 | -2.47838891 | 1 | uM |
| QL-X-138 | BCWM.1 | IRE1 | DLKPHNILISMPNAHGK | Lys2 | 5.339267666 | 1 | uM |
| QL-X-138 | BCWM.1 | ITPK1 | ESIFFNSHNVSKPESSSVLTELDKIEGVFERPSDEVIR | ATP | 34.13986871 | 1 | uM |
| QL-X-138 | BCWM.1 | JAK1_domain2 | IGDFGLTKAIETDKEYYTVK | Activation Loop | 60.68936501 | 1 | uM |