QL-X-138 KiNativ -- single dose experiment - Dataset (ID:20204)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-X-138 | BCWM.1 | JAK3 domain2 | IADFGLAKLLPLDKDYYVVR | Activation Loop | 60.82830234 | 1 | uM |
| QL-X-138 | BCWM.1 | JNK1,JNK2,JNK3 | DLKPSNIVVK | Lys2 | 13.40506031 | 1 | uM |
| QL-X-138 | BCWM.1 | KHS1 | NVHTGELAAVKIIK | Lys1 | -0.477114387 | 1 | uM |
| QL-X-138 | BCWM.1 | KSR1,KSR2 | SKNVFYDNGK | Activation Loop | 8.27219181 | 1 | uM |
| QL-X-138 | BCWM.1 | LATS1 | ALYATKTLR | Lys1 | 26.42303305 | 1 | uM |
| QL-X-138 | BCWM.1 | LATS2 | DIKPDNILIDLDGHIK | Lys2 | 28.03028261 | 1 | uM |
| QL-X-138 | BCWM.1 | LKB1 | DIKPGNLLLTTGGTLK | Lys2 | 14.63647065 | 1 | uM |
| QL-X-138 | BCWM.1 | LOK | DLKAGNVLMTLEGDIR | Lys2 | -21.24010057 | 1 | uM |
| QL-X-138 | BCWM.1 | LRRK2 | DLKPHNVLLFTLYPNAAIIAK | Lys2 | 45.4508605 | 1 | uM |
| QL-X-138 | BCWM.1 | LYN | VAVKTLKPGTMSVQAFLEEANLMK | Lys1 | 61.37351181 | 1 | uM |
| QL-X-138 | BCWM.1 | MAP2K1,MAP2K2 | DVKPSNILVNSR | Lys2 | 7.910761282 | 1 | uM |
| QL-X-138 | BCWM.1 | MAP2K3 | DVKPSNVLINK | Lys2 | 8.464981447 | 1 | uM |
| QL-X-138 | BCWM.1 | MAP2K4 | DIKPSNILLDR | Lys2 | 8.146709089 | 1 | uM |
| QL-X-138 | BCWM.1 | MAP2K5 | DVKPSNMLVNTR | Lys2 | -9.160888835 | 1 | uM |
| QL-X-138 | BCWM.1 | MAP2K6 | DVKPSNVLINALGQVK | Lys2 | -39.73473579 | 1 | uM |
| QL-X-138 | BCWM.1 | MP2K7 | DVKPSNILLDER | Lys2 | -4.523234116 | 1 | uM |
| QL-X-138 | BCWM.1 | MAP3K1 | DVKGANLLIDSTGQR | Lys2 | 2.793987227 | 1 | uM |
| QL-X-138 | BCWM.1 | M3K2,MAP3K3 | DIKGANILR | Lys2 | 6.564957339 | 1 | uM |
| QL-X-138 | BCWM.1 | MAP3K4 | DIKGANIFLTSSGLIK | Lys2 | -12.17088834 | 1 | uM |
| QL-X-138 | BCWM.1 | MAP3K5 | DIKGDNVLINTYSGVLK | Lys2 | 0.729091186 | 1 | uM |
| QL-X-138 | BCWM.1 | MARK3 | EVAIKIIDKTQLNPTSLQK | Lys1 | 45.65066563 | 1 | uM |
| QL-X-138 | BCWM.1 | MARK3,MARK4 | EVAIKIIDK | Lys1 | 3.114402142 | 1 | uM |
| QL-X-138 | BCWM.1 | MAST1,MAST2 | DLKPDNLLITSMGHIK | Lys2 | 44.6017691 | 1 | uM |
| QL-X-138 | BCWM.1 | MAST3 | DLKPDNLLITSLGHIK | Lys2 | 38.94230574 | 1 | uM |
| QL-X-138 | BCWM.1 | MASTL | GAFGKVYLGQK | ATP Loop | -0.462372082 | 1 | uM |