QL-X-138 KiNativ -- single dose experiment - Dataset (ID:20204)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
QL-X-138 BCWM.1 FRK
HEIKLPVK
Activation Loop
0.087392973
1
uM
QL-X-138 BCWM.1 KSR1
SKNVFYDNGKVVITDFGLFGISGVVR
Activation Loop
52.54874503
1
uM
QL-X-138 BCWM.1 LCK
EGAKFPIKWTAPEAINYGTFTIK
Activation Loop
26.15622742
1
uM
QL-X-138 BCWM.1 NEK2
DLKPANVFLDGK
Lys2
6.565871129
1
uM
QL-X-138 BCWM.1 STK33
DLKLENIMVK
Lys2
34.78219334
1
uM
QL-X-138 BCWM.1 TYK2(Kin.Dom.2)
IGDFGLAKAVPEGHEYYR
Activation Loop
13.07024614
1
uM
QL-X-138 BCWM.1 Wnk1,Wnk2
GSFKTVYK
ATP Loop
-1.126339473
1
uM
QL-X-138 BCWM.1 MER,TYRO3
KIYSGDYYR
Activation Loop
3.734337363
1
uM
QL-X-138 BCWM.1 RSK2 domain1
DLKPENILLDEEGHIKLTDFGLSKESIDHEK
Lys2
32.51384261
1
uM