QL-X-138 KiNativ -- single dose experiment - Dataset (ID:20204)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| QL-X-138 | BCWM.1 | ABL,ARG | LMTGDTYTAHAGAKFPIK | Activation Loop | 25.73794561 | 1 | uM |
| QL-X-138 | BCWM.1 | AMPKa1,AMPKa2 | DLKPENVLLDAHMNAK | Lys2 | 29.49947815 | 1 | uM |
| QL-X-138 | BCWM.1 | ARAF | DLKSNNIFLHEGLTVK | Lys2 | 57.4717555 | 1 | uM |
| QL-X-138 | BCWM.1 | ATR | FYIMMCKPK | ATP | 78.07794049 | 1 | uM |
| QL-X-138 | BCWM.1 | AurA | FILALKVLFK | Lys1 | 74.00960491 | 1 | uM |
| QL-X-138 | BCWM.1 | AurB | SHFIVALKVLFK | Lys1 | 35.98896891 | 1 | uM |
| QL-X-138 | BCWM.1 | BARK1 | DLKPANILLDEHGHVR | Lys2 | 10.63576754 | 1 | uM |
| QL-X-138 | BCWM.1 | BRAF | DLKSNNIFLHEDLTVK | Lys2 | 63.68312741 | 1 | uM |
| QL-X-138 | BCWM.1 | BTK | YVLDDEYTSSVGSKFPVR | Activation Loop | >99 | 1 | uM |
| QL-X-138 | BCWM.1 | CaMK1a | LVAIKCIAK | Lys1 | -27.71597238 | 1 | uM |
| QL-X-138 | BCWM.1 | CAMK1D | LFAVKCIPK | Lys1 | 7.981646566 | 1 | uM |
| QL-X-138 | BCWM.1 | CaMK2g | TSTQEYAAKIINTK | Lys1 | -15.78345401 | 1 | uM |
| QL-X-138 | BCWM.1 | CaMKK2 | DIKPSNLLVGEDGHIK | Lys2 | 9.712956785 | 1 | uM |
| QL-X-138 | BCWM.1 | CASK | ETGQQFAVKIVDVAK | Lys1 | 13.79525009 | 1 | uM |
| QL-X-138 | BCWM.1 | CDC2 | DLKPQNLLIDDKGTIK | Lys2 | 7.249150054 | 1 | uM |
| QL-X-138 | BCWM.1 | CDK11,CDK8 | DLKPANILVMGEGPER | Lys2 | 18.2342496 | 1 | uM |
| QL-X-138 | BCWM.1 | CDK2 | DLKPQNLLINTEGAIK | Lys2 | -8.525927163 | 1 | uM |
| QL-X-138 | BCWM.1 | CDK4 | DLKPENILVTSGGTVK | Lys2 | 6.738395305 | 1 | uM |
| QL-X-138 | BCWM.1 | CDK5 | DLKPQNLLINR | Lys2 | -5.292754551 | 1 | uM |
| QL-X-138 | BCWM.1 | CDK6 | DLKPQNILVTSSGQIK | Lys2 | -24.10699447 | 1 | uM |
| QL-X-138 | BCWM.1 | CDK7 | DLKPNNLLLDENGVLK | Lys2 | -4.444192192 | 1 | uM |
| QL-X-138 | BCWM.1 | CDK9 | DMKAANVLITR | Lys2 | -1.851232927 | 1 | uM |
| QL-X-138 | BCWM.1 | CHK2 | DLKPENVLLSSQEEDCLIK | Lys2 | 75.84872918 | 1 | uM |
| QL-X-138 | BCWM.1 | KC1A | DIKPDNFLMGIGR | Lys2 | 14.057419 | 1 | uM |
| QL-X-138 | BCWM.1 | CLK3 | YEIVGNLGEGTFGKVVECLDHAR | ATP Loop | 25.53508914 | 1 | uM |