VX-680 KINOMEscan - Dataset (ID:20197)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Tozasertib | KIT | 240.0 | nM |
| Tozasertib | KIT(A829P) | 380.0 | nM |
| Tozasertib | KIT(D816H) | 1900.0 | nM |
| Tozasertib | KIT(D816V) | 290.0 | nM |
| Tozasertib | KIT(L576P) | 230.0 | nM |
| Tozasertib | KIT(V559D) | 240.0 | nM |
| Tozasertib | KIT(V559D,T670I) | 430.0 | nM |
| Tozasertib | KIT(V559D,V654A) | 2300.0 | nM |
| Tozasertib | LATS1 | 5500.0 | nM |
| Tozasertib | LATS2 | 6500.0 | nM |
| Tozasertib | LCK | 61.0 | nM |
| Tozasertib | LIMK1 | 2600.0 | nM |
| Tozasertib | LIMK2 | 2600.0 | nM |
| Tozasertib | LKB1 | 1300.0 | nM |
| Tozasertib | LOK | 120.0 | nM |
| Tozasertib | LRRK2 | nM | |
| Tozasertib | LRRK2(G2019S) | nM | |
| Tozasertib | LTK | 7500.0 | nM |
| Tozasertib | LYN | 650.0 | nM |
| Tozasertib | M3K13 | 180.0 | nM |
| Tozasertib | MAK | nM | |
| Tozasertib | MAP3K1 | nM | |
| Tozasertib | MAP3K15 | nM | |
| Tozasertib | M3K2 | 1100.0 | nM |
| Tozasertib | MAP3K3 | 1900.0 | nM |