VX-680 KINOMEscan - Dataset (ID:20197)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Tozasertib | MAP3K4 | 2500.0 | nM |
Tozasertib | MAP4K2 | 2600.0 | nM |
Tozasertib | M4K3 | 290.0 | nM |
Tozasertib | MAP4K4 | 2400.0 | nM |
Tozasertib | MAP4K5 | 83.0 | nM |
Tozasertib | MAPKAPK2 | 3800.0 | nM |
Tozasertib | MAPKAPK5 | nM | |
Tozasertib | MARK1 | 4900.0 | nM |
Tozasertib | MARK2 | 1400.0 | nM |
Tozasertib | MARK3 | 2500.0 | nM |
Tozasertib | MARK4 | 4900.0 | nM |
Tozasertib | MAST1 | nM | |
Tozasertib | MP2K1 | 1800.0 | nM |
Tozasertib | MP2K2 | 2000.0 | nM |
Tozasertib | MP2K3 | nM | |
Tozasertib | MP2K4 | nM | |
Tozasertib | MP2K5 | 260.0 | nM |
Tozasertib | MP2K6 | 2600.0 | nM |
Tozasertib | MELK | 240.0 | nM |
Tozasertib | MERTK | 1700.0 | nM |
Tozasertib | MET | 670.0 | nM |
Tozasertib | MET(M1250T) | 480.0 | nM |
Tozasertib | MET(Y1235D) | 360.0 | nM |
Tozasertib | MINK | 1100.0 | nM |
Tozasertib | MP2K7 | nM |