VX-680 KINOMEscan - Dataset (ID:20197)

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Small Molecule Protein Kd Conc unit
Tozasertib MAP3K4 2500.0
nM
Tozasertib MAP4K2 2600.0
nM
Tozasertib M4K3 290.0
nM
Tozasertib MAP4K4 2400.0
nM
Tozasertib MAP4K5 83.0
nM
Tozasertib MAPKAPK2 3800.0
nM
Tozasertib MAPKAPK5
nM
Tozasertib MARK1 4900.0
nM
Tozasertib MARK2 1400.0
nM
Tozasertib MARK3 2500.0
nM
Tozasertib MARK4 4900.0
nM
Tozasertib MAST1
nM
Tozasertib MP2K1 1800.0
nM
Tozasertib MP2K2 2000.0
nM
Tozasertib MP2K3
nM
Tozasertib MP2K4
nM
Tozasertib MP2K5 260.0
nM
Tozasertib MP2K6 2600.0
nM
Tozasertib MELK 240.0
nM
Tozasertib MERTK 1700.0
nM
Tozasertib MET 670.0
nM
Tozasertib MET(M1250T) 480.0
nM
Tozasertib MET(Y1235D) 360.0
nM
Tozasertib MINK 1100.0
nM
Tozasertib MP2K7
nM