VX-680 KINOMEscan - Dataset (ID:20197)

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Small Molecule Protein Kd Conc unit
Tozasertib MKNK1
nM
Tozasertib MKNK2 5200.0
nM
Tozasertib MLCK 15.0
nM
Tozasertib MLK1 390.0
nM
Tozasertib MLK2 1800.0
nM
Tozasertib MLK3 680.0
nM
Tozasertib MRCKA
nM
Tozasertib MRCKB
nM
Tozasertib MST1 200.0
nM
Tozasertib MST1R 1300.0
nM
Tozasertib MST2 510.0
nM
Tozasertib MST3 3600.0
nM
Tozasertib MST4 3500.0
nM
Tozasertib MTOR
nM
Tozasertib MUSK 300.0
nM
Tozasertib MYLK
nM
Tozasertib MYLK2 43.0
nM
Tozasertib MYLK4 2200.0
nM
Tozasertib MYO3A
nM
Tozasertib MYO3B
nM
Tozasertib NDR1
nM
Tozasertib NDR2 6900.0
nM
Tozasertib NEK1
nM
Tozasertib NEK11
nM
Tozasertib NEK2
nM