VX-680 KINOMEscan - Dataset (ID:20197)
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Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Tozasertib | HCK | 6200.0 | nM |
Tozasertib | HIPK1 | nM | |
Tozasertib | HIPK2 | nM | |
Tozasertib | HIPK3 | nM | |
Tozasertib | HIPK4 | nM | |
Tozasertib | M4K1 | 72.0 | nM |
Tozasertib | HUNK | 9800.0 | nM |
Tozasertib | ICK | nM | |
Tozasertib | IGF1R | 740.0 | nM |
Tozasertib | IKKA | nM | |
Tozasertib | IKKB | nM | |
Tozasertib | IKKE | 2600.0 | nM |
Tozasertib | INSR | 630.0 | nM |
Tozasertib | INSRR | 290.0 | nM |
Tozasertib | IRAK1 | nM | |
Tozasertib | IRAK3 | nM | |
Tozasertib | IRAK4 | 3700.0 | nM |
Tozasertib | ITK | 350.0 | nM |
Tozasertib | JAK1(JH1domain-catalytic) | 5900.0 | nM |
Tozasertib | JAK1(JH2domain-pseudokinase) | nM | |
Tozasertib | JAK2(JH1domain-catalytic) | 190.0 | nM |
Tozasertib | JAK3(JH1domain-catalytic) | 630.0 | nM |
Tozasertib | JNK1 | nM | |
Tozasertib | MK09 | nM | |
Tozasertib | JNK3 | 2800.0 | nM |