VX-680 KINOMEscan - Dataset (ID:20197)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Tozasertib | RSK2(Kin.Dom.1-N-terminal) | 6400.0 | nM |
Tozasertib | RSK3(Kin.Dom.1-N-terminal) | 2000.0 | nM |
Tozasertib | RSK3(Kin.Dom.2-C-terminal) | nM | |
Tozasertib | RSK4(Kin.Dom.1-N-terminal) | nM | |
Tozasertib | RSK4(Kin.Dom.2-C-terminal) | nM | |
Tozasertib | S6K1 | nM | |
Tozasertib | SBK1 | nM | |
Tozasertib | SgK110 | 530.0 | nM |
Tozasertib | SGK3 | nM | |
Tozasertib | SIK1 | 2500.0 | nM |
Tozasertib | SIK2 | 1700.0 | nM |
Tozasertib | SLK | 82.0 | nM |
Tozasertib | SNARK | 530.0 | nM |
Tozasertib | SNRK | nM | |
Tozasertib | SRC | 170.0 | nM |
Tozasertib | SRMS | nM | |
Tozasertib | SRPK1 | 82.0 | nM |
Tozasertib | SRPK2 | 680.0 | nM |
Tozasertib | SRPK3 | 240.0 | nM |
Tozasertib | STK16 | 610.0 | nM |
Tozasertib | STK33 | nM | |
Tozasertib | STK35 | nM | |
Tozasertib | STK36 | nM | |
Tozasertib | STK39 | nM | |
Tozasertib | SYK | 1800.0 | nM |