VX-680 KINOMEscan - Dataset (ID:20197)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Tozasertib | EPHA1 | 1000.0 | nM |
Tozasertib | EPHA2 | 840.0 | nM |
Tozasertib | EPHA3 | 1500.0 | nM |
Tozasertib | EPHA4 | 4300.0 | nM |
Tozasertib | EPHA5 | nM | |
Tozasertib | EPHA6 | 4700.0 | nM |
Tozasertib | EPHA7 | nM | |
Tozasertib | EPHA8 | 500.0 | nM |
Tozasertib | EPHB1 | 1900.0 | nM |
Tozasertib | EPHB2 | 5600.0 | nM |
Tozasertib | EPHB3 | nM | |
Tozasertib | EPHB4 | 1700.0 | nM |
Tozasertib | EPHB6 | 28.0 | nM |
Tozasertib | ERBB2 | nM | |
Tozasertib | ERBB3 | 7100.0 | nM |
Tozasertib | ERBB4 | nM | |
Tozasertib | MK03 | nM | |
Tozasertib | MK01 | nM | |
Tozasertib | ERK3 | nM | |
Tozasertib | ERK4 | nM | |
Tozasertib | ERK5 | 6800.0 | nM |
Tozasertib | ERK8 | nM | |
Tozasertib | ERN1 | 5600.0 | nM |
Tozasertib | FAK1 | nM | |
Tozasertib | FER | 4200.0 | nM |