VX-680 KINOMEscan - Dataset (ID:20197)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | Kd | Conc unit |
---|---|---|---|
Tozasertib | TAK1 | 2300.0 | nM |
Tozasertib | TAOK1 | 290.0 | nM |
Tozasertib | TAOK2 | 430.0 | nM |
Tozasertib | TAOK3 | 81.0 | nM |
Tozasertib | TBK1 | 490.0 | nM |
Tozasertib | TEC | 8700.0 | nM |
Tozasertib | TESK1 | 5600.0 | nM |
Tozasertib | TGFBR1 | 8400.0 | nM |
Tozasertib | TGFBR2 | nM | |
Tozasertib | TIE1 | 270.0 | nM |
Tozasertib | TIE2 | 450.0 | nM |
Tozasertib | TLK1 | 4000.0 | nM |
Tozasertib | TLK2 | nM | |
Tozasertib | TNIK | 1800.0 | nM |
Tozasertib | TNK1 | 83.0 | nM |
Tozasertib | TNK2 | 4400.0 | nM |
Tozasertib | TNNI3K | nM | |
Tozasertib | TRKA | 38.0 | nM |
Tozasertib | TRKB | 240.0 | nM |
Tozasertib | TRKC | 200.0 | nM |
Tozasertib | TRPM6 | nM | |
Tozasertib | TSSK1 | nM | |
Tozasertib | TTK | 8100.0 | nM |
Tozasertib | TXK | 2700.0 | nM |
Tozasertib | TYK2(JH1domain-catalytic) | 510.0 | nM |