TG-101348 KINOMEscan - Dataset (ID:20174)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Fedratinib | KIT | 130.0 | nM |
| Fedratinib | KIT(A829P) | 46.0 | nM |
| Fedratinib | KIT(D816H) | 160.0 | nM |
| Fedratinib | KIT(D816V) | 160.0 | nM |
| Fedratinib | KIT(L576P) | 120.0 | nM |
| Fedratinib | KIT(V559D) | 58.0 | nM |
| Fedratinib | KIT(V559D,T670I) | 1500.0 | nM |
| Fedratinib | KIT(V559D,V654A) | 3500.0 | nM |
| Fedratinib | LATS1 | nM | |
| Fedratinib | LATS2 | 8000.0 | nM |
| Fedratinib | LCK | 72.0 | nM |
| Fedratinib | LIMK1 | 940.0 | nM |
| Fedratinib | LIMK2 | 7900.0 | nM |
| Fedratinib | LKB1 | 310.0 | nM |
| Fedratinib | LOK | 2900.0 | nM |
| Fedratinib | LRRK2 | 870.0 | nM |
| Fedratinib | LRRK2(G2019S) | 1000.0 | nM |
| Fedratinib | LTK | 6300.0 | nM |
| Fedratinib | LYN | 500.0 | nM |
| Fedratinib | M3K13 | 590.0 | nM |
| Fedratinib | MAK | nM | |
| Fedratinib | MAP3K1 | nM | |
| Fedratinib | MAP3K15 | nM | |
| Fedratinib | M3K2 | 580.0 | nM |
| Fedratinib | MAP3K3 | 1300.0 | nM |