TG-101348 KINOMEscan - Dataset (ID:20174)

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Small Molecule Protein Kd Conc unit
Fedratinib MAP3K4 4100.0
nM
Fedratinib MAP4K2 2100.0
nM
Fedratinib M4K3 1800.0
nM
Fedratinib MAP4K4
nM
Fedratinib MAP4K5
nM
Fedratinib MAPKAPK2
nM
Fedratinib MAPKAPK5
nM
Fedratinib MARK1 700.0
nM
Fedratinib MARK2 3100.0
nM
Fedratinib MARK3 300.0
nM
Fedratinib MARK4 970.0
nM
Fedratinib MAST1
nM
Fedratinib MP2K1 5100.0
nM
Fedratinib MP2K2 3100.0
nM
Fedratinib MP2K3 3500.0
nM
Fedratinib MP2K4 9900.0
nM
Fedratinib MP2K5 360.0
nM
Fedratinib MP2K6
nM
Fedratinib MELK 2600.0
nM
Fedratinib MERTK 820.0
nM
Fedratinib MET 8500.0
nM
Fedratinib MET(M1250T) 4400.0
nM
Fedratinib MET(Y1235D)
nM
Fedratinib MINK 8900.0
nM
Fedratinib MP2K7
nM