TG-101348 KINOMEscan - Dataset (ID:20174)
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| Small Molecule | Protein | Kd | Conc unit |
|---|---|---|---|
| Fedratinib | HCK | 2100.0 | nM |
| Fedratinib | HIPK1 | 860.0 | nM |
| Fedratinib | HIPK2 | 1000.0 | nM |
| Fedratinib | HIPK3 | 1300.0 | nM |
| Fedratinib | HIPK4 | 220.0 | nM |
| Fedratinib | M4K1 | 1300.0 | nM |
| Fedratinib | HUNK | nM | |
| Fedratinib | ICK | 1900.0 | nM |
| Fedratinib | IGF1R | 2200.0 | nM |
| Fedratinib | IKKA | 830.0 | nM |
| Fedratinib | IKKB | 360.0 | nM |
| Fedratinib | IKKE | 360.0 | nM |
| Fedratinib | INSR | 850.0 | nM |
| Fedratinib | INSRR | 1600.0 | nM |
| Fedratinib | IRAK1 | 220.0 | nM |
| Fedratinib | IRAK3 | 120.0 | nM |
| Fedratinib | IRAK4 | 1200.0 | nM |
| Fedratinib | ITK | 490.0 | nM |
| Fedratinib | JAK1(JH1domain-catalytic) | 18.0 | nM |
| Fedratinib | JAK1(JH2domain-pseudokinase) | 2000.0 | nM |
| Fedratinib | JAK2(JH1domain-catalytic) | 1.1 | nM |
| Fedratinib | JAK3(JH1domain-catalytic) | 74.0 | nM |
| Fedratinib | JNK1 | 260.0 | nM |
| Fedratinib | MK09 | 240.0 | nM |
| Fedratinib | JNK3 | 200.0 | nM |