NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
-9.9
0.05
uM
NVP-BHG712 PC-3 YANK3
DVkPDNILLDER
Lys2
4.4
0.05
uM
NVP-BHG712 PC-3 MLTK
WISQDKEVAVKk
Lys1
49.9
0.05
uM
NVP-BHG712 PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
7.8
0.05
uM