NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

 Full screen view
Filter results: >>>>
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 FYV1
GGkSGAAFYATEDDRFILK
ATP
14.1
 0.05
uM
NVP-BHG712 PC-3 PITSLRE
DLkTSNLLLSHAGILK
Lys2
2.8
 0.05
uM
NVP-BHG712 PC-3 PRKACB
DLkPENLLIDHQGYIQ
Lys2
-8.0
 0.05
uM
NVP-BHG712 PC-3 PKD3
NIVHCDLkPENVLLASAEPFPQVK
Lys2
-20.7
 0.05
uM
NVP-BHG712 PC-3 PKN1
VLLSEFRPSGELFAIkALK
Lys1
-14.4
 0.05
uM
NVP-BHG712 PC-3 PKN2
DLkLDNLLLDTEGFVK
Lys2
13.0
 0.05
uM
NVP-BHG712 PC-3 PKR
DLkPSNIFLVDTK
Lys2
-3.2
 0.05
uM
NVP-BHG712 PC-3 PLK1
CFEISDADTKEVFAGkIVPK
Lys1
-12.5
 0.05
uM
NVP-BHG712 PC-3 PLK1
DLkLGNLFLNEDLEVK
Lys2
10.3
 0.05
uM
NVP-BHG712 PC-3 PRP4
CNILHADIkPDNILVNESK
Lys2
0.2
 0.05
uM
NVP-BHG712 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
30.6
 0.05
uM
NVP-BHG712 PC-3 QIK
TEVAIkIIDK
Lys1
3.4
 0.05
uM
NVP-BHG712 PC-3 RAF1
DMkSNNIFLHEGLTVK
Lys2
-13.4
 0.05
uM
NVP-BHG712 PC-3 RIPK2
VQVAVkHLHIHTPLLDSER
Lys1
-3.5
 0.05
uM
NVP-BHG712 PC-3 ROCK1
kLQLELNQER
Other
-8.0
 0.05
uM
NVP-BHG712 PC-3 ROCK1,ROCK2
DVkPDNMLLDK
Lys2
-18.5
 0.05
uM
NVP-BHG712 PC-3 RON
IQCAIkSLSR
Lys1
1.5
 0.05
uM
NVP-BHG712 PC-3 RSK1_domain2
DLkPSNILYVDESGNPECLR
Lys2
-8.3
 0.05
uM
NVP-BHG712 PC-3 RSK1,RSK2_domain1
DLkPENILLDEEGHIKLTDFGLSK
Lys2
-2.7
 0.05
uM
NVP-BHG712 PC-3 RSK1,RSK2,RSK3_domain1
DLkPENILLDEEGHIK
Lys2
7.0
 0.05
uM
NVP-BHG712 PC-3 RSK1,RSK3_domain2
SkRDPSEEIEILLR
Protein Kinase Domain
-1.8
 0.05
uM
NVP-BHG712 PC-3 RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
-9.3
 0.05
uM
NVP-BHG712 PC-3 RSK2 domain1
VLGQGSFGkVFLVK
ATP Loop
3.0
 0.05
uM
NVP-BHG712 PC-3 RSK2_domain2
DLkPSNILYVDESGNPESIR
Lys2
-0.4
 0.05
uM
NVP-BHG712 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
-16.0
 0.05
uM