NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| NVP-BHG712 | PC-3 | OSR1 | DVkAGNILLGEDGSVQIADFGVSAFLATGGDITR | Lys2 | -6.2 | 0.05 | uM |
| NVP-BHG712 | PC-3 | p38a | DLkPSNLAVNEDCELK | Lys2 | 61.0 | 0.05 | uM |
| NVP-BHG712 | PC-3 | MK14 | QELNkTIWEVPER | Other | 26.8 | 0.05 | uM |
| NVP-BHG712 | PC-3 | MK11 | QELNkTVWEVPQR | Other | -24.1 | 0.05 | uM |
| NVP-BHG712 | PC-3 | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | 1.1 | 0.05 | uM |
| NVP-BHG712 | PC-3 | KS6B1 | DLkPENIMLNHQGHVK | Lys2 | -17.0 | 0.05 | uM |
| NVP-BHG712 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | 1.6 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK16 | LTDNLVALkEIR | Lys1 | 7.3 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PCTAIRE2 | DLkPQNLLINEK | Lys2 | -7.4 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PCTAIRE2,PCTAIRE3 | SKLTENLVALkEIR | Lys1 | -13.2 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PEK | DLkPSNIFFTMDDVVK | Lys2 | 7.8 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK14 | LVALkVIR | Lys1 | -8.7 | 0.05 | uM |
| NVP-BHG712 | PC-3 | CDK14 | DLkPQNLLISDTGELK | Lys2 | 0.9 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PHKg1 | DLkPENILLDDNMNIK | Lys2 | 1.9 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | -21.2 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 2.1 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PI4KB | VPHTQAVVLNSkDKAPYLIYVEVLECENFDTTSVPAR | ATP | -14.1 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PIK3C3 | TEDGGKYPVIFkHGDDLRQDQLILQIISLMDK | ATP | 7.0 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PIK3C3 | TEDGGKYPVIFkHGDDLR | ATP | -5.7 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | -3.4 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PIP4K2A | AKELPTLkDNDFINEGQK | ATP | -3.4 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PIP4K2B | DLPTFkDNDFLNEGQK | ATP | 26.7 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PI42C | VKELPTLkDMDFLNK | ATP | -14.7 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PI42C | ELPTLkDMDFLNK | ATP | 1.2 | 0.05 | uM |
| NVP-BHG712 | PC-3 | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | -7.4 | 0.05 | uM |