NVP-BHG712 KiNativ -- multiple dose experiment - Dataset (ID:20104)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
NVP-BHG712 PC-3 MARK3,MARK4
EVAIkIIDK
Lys1
-9.3
 0.50
uM
NVP-BHG712 PC-3 MAST1,MAST2
DLkPDNLLITSMGHIK
Lys2
-22.0
 0.50
uM
NVP-BHG712 PC-3 MAST2,MAST4
DLkPDNLLVTSMGHIK
Lys2
0.6
 0.50
uM
NVP-BHG712 PC-3 MAST3
DLkPDNLLITSLGHIK
Lys2
0.5
 0.50
uM
NVP-BHG712 PC-3 MASTL
GAFGkVYLGQK
ATP Loop
3.5
 0.50
uM
NVP-BHG712 PC-3 MET
DMYDkEYYSVHNK
Activation Loop
14.4
 0.50
uM
NVP-BHG712 PC-3 MLK1,MLKL
DLkSSNILILQK
Lys2
7.1
 0.50
uM
NVP-BHG712 PC-3 MLK3
DLkSNNILLLQPIESDDMEHK
Lys2
9.5
 0.50
uM
NVP-BHG712 PC-3 MLK4
DLkSSNILLLEK
Lys2
13.1
 0.50
uM
NVP-BHG712 PC-3 MLKL
APVAIkVFK
Lys1
9.9
 0.50
uM
NVP-BHG712 PC-3 MRCKb
DIkPDNVLLDVNGHIR
Lys2
-2.0
 0.50
uM
NVP-BHG712 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
-11.7
 0.50
uM
NVP-BHG712 PC-3 MSK1 domain1
LGIIYRDIkLENILLDSNGHVVLTDFGLSK
Lys2
7.0
 0.50
uM
NVP-BHG712 PC-3 MSK1_domain1
DIkLENILLDSNGHVVLTDFGLSK
Lys2
3.3
 0.50
uM
NVP-BHG712 PC-3 MSK1,MSK2_domain1
VLGTGAYGkVFLVR
ATP Loop
2.5
 0.50
uM
NVP-BHG712 PC-3 MSK2 domain1
DLkLENVLLDSEGHIVLTDFGLSK
Lys2
4.6
 0.50
uM
NVP-BHG712 PC-3 MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
14.3
 0.50
uM
NVP-BHG712 PC-3 MST1,MST2
DIkAGNILLNTEGHAK
Lys2
9.6
 0.50
uM
NVP-BHG712 PC-3 MST2
ESGQVVAIkQVPVESDLQEIIK
Lys1
6.7
 0.50
uM
NVP-BHG712 PC-3 MST3
DIkAANVLLSEHGEVK
Lys2
5.3
 0.50
uM
NVP-BHG712 PC-3 MST4,YSK1
DIkAANVLLSEQGDVK
Lys2
12.2
 0.50
uM
NVP-BHG712 PC-3 NDR1
DTGHVYAMkILR
Lys1
-24.8
 0.50
uM
NVP-BHG712 PC-3 NDR2
DTGHIYAMkILR
Lys1
-16.6
 0.50
uM
NVP-BHG712 PC-3 NDR2
DIkPDNLLLDAK
Lys2
-2.1
 0.50
uM
NVP-BHG712 PC-3 NEK1
DIkSQNIFLTK
Lys2
3.9
 0.50
uM