XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 HeLa TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
-28.1
10
uM
XMD8-92 PC-3 TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
5.6
10
uM
XMD8-92 PC-3 TAOK2
DVkAGNILLSEPGLVK
Lys2
5.6
10
uM
XMD8-92 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
-43.4
10
uM
XMD8-92 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
6.9
10
uM
XMD8-92 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
3.4
10
uM
XMD8-92 PC-3 TLK2
YVAVkIHQLNK
Lys1
7.8
10
uM
XMD8-92 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
-6.2
10
uM
XMD8-92 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
-10.4
10
uM
XMD8-92 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-1.9
10
uM
XMD8-92 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
8.8
10
uM
XMD8-92 HeLa MLTK
WISQDKEVAVKk
Lys1
-0.8
10
uM
XMD8-92 PC-3 MLTK
WISQDKEVAVKk
Lys1
10.9
10
uM
XMD8-92 HeLa ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-24.3
10
uM
XMD8-92 PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
0.5
10
uM
XMD8-92 HeLa BARK1
DLkPANILLDEHGHVR
Lys2
9.3
10
uM
XMD8-92 HeLa BTK
GQYDVAIkMIK
Lys1
-9.2
10
uM
XMD8-92 HeLa CAMK1D
LFAVkCIPK
Lys1
-3.6
10
uM
XMD8-92 PC-3 CDK5
DLkPQNLLINR
Lys2
-1.0
10
uM
XMD8-92 HeLa CHK1
DIkPENLLLDER
Lys2
1.3
10
uM
XMD8-92 HeLa CHK2
DLkPENVLLSSQEEDCLIK
Lys2
-1.4
10
uM
XMD8-92 PC-3 CHK2
DLkPENVLLSSQEEDCLIK
Lys2
8.3
10
uM
XMD8-92 HeLa DGKA
IDPVPNTHPLLVFVNPkSGGK
ATP
-25.7
10
uM
XMD8-92 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
-3.7
10
uM
XMD8-92 HeLa FES
LRADNTLVAVkSCR
Lys1
-4.8
10
uM