XMD8-92 KiNativ -- single dose experiment - Dataset (ID:20102)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-92 PC-3 PI4KB
VPHTQAVVLNSkDK
ATP
7.0
 10
uM
XMD8-92 HeLa PIK3C3
TEDGGKYPVIFkHGDDLR
ATP
4.9
 10
uM
XMD8-92 PC-3 PIK3CB
VFGEDSVGVIFkNGDDLRQDMLTLQMLR
ATP
-69.6
 10
uM
XMD8-92 HeLa PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
3.6
 10
uM
XMD8-92 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
10.9
 10
uM
XMD8-92 PC-3 PITSLRE
DLkTSNLLLSHAGILK
Lys2
1.6
 10
uM
XMD8-92 PC-3 PKCa,PKCb
DLkLDNVMLDSEGHIK
Lys2
-12.7
 10
uM
XMD8-92 HeLa PKD1,PKD2
NIVHCDLkPENVLLASADPFPQVK
Lys2
4.2
 10
uM
XMD8-92 HeLa PKR
DLkPSNIFLVDTK
Lys2
-11.5
 10
uM
XMD8-92 PC-3 PKR
DLkPSNIFLVDTK
Lys2
4.6
 10
uM
XMD8-92 HeLa PRPK
FLSGLELVkQGAEAR
ATP Loop
-2.4
 10
uM
XMD8-92 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
9.7
 10
uM
XMD8-92 PC-3 ROCK1,ROCK2
DVkPDNMLLDK
Lys2
-11.0
 10
uM
XMD8-92 HeLa RSK1,RSK2_domain1
DLkPENILLDEEGHIKLTDFGLSK
Lys2
30.3
 10
uM
XMD8-92 HeLa RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
-2.5
 10
uM
XMD8-92 PC-3 RSK2_domain2
DLkPSNILYVDESGNPESIR
Lys2
27.9
 10
uM
XMD8-92 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
-9.2
 10
uM
XMD8-92 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
22.4
 10
uM
XMD8-92 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
-20.2
 10
uM
XMD8-92 HeLa SGK3
FYAVkVLQK
Lys1
-8.8
 10
uM
XMD8-92 HeLa SLK
DLkAGNILFTLDGDIK
Lys2
-6.5
 10
uM
XMD8-92 PC-3 SLK
DLkAGNILFTLDGDIK
Lys2
4.3
 10
uM
XMD8-92 HeLa SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
6.4
 10
uM
XMD8-92 PC-3 SRC
VAIkTLKPGTMSPEAFLQEAQVMK
Lys1
17.5
 10
uM
XMD8-92 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
-20.9
 10
uM